Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50004424
LigandPNGBDBM50482773(CHEMBL1253513)
Affinity DataKi:  1.92E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482766(CHEMBL1254501)
Affinity DataKi:  2.08E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482769(CHEMBL1253486)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482770(CHEMBL1253511)
Affinity DataKi:  3.64E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50086502(2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole | 2-BFi...)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482764(CHEMBL1254500)
Affinity DataKi:  4.39E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482768(CHEMBL1254502)
Affinity DataKi:  4.43E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482767(CHEMBL1253584)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482765(CHEMBL1253512)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482771(CHEMBL1253583)
Affinity DataKi:  2.42E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
LigandPNGBDBM50482772(CHEMBL1253510)
Affinity DataKi:  2.55E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2 adrenergic receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed