Compile Data Set for Download or QSAR
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Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50039312
Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330441(3-amino-2-(4-(4-(quinolin-2-yl)piperazin-1-yl)buty...)
Affinity DataKi:  4.72nMAssay Description:Binding affinity to human 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330444(3-Amino-7-nitro-2-[3-(4-quinolin-2-ylpiperazin-1-y...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330441(3-amino-2-(4-(4-(quinolin-2-yl)piperazin-1-yl)buty...)
Affinity DataIC50: >1.40nMAssay Description:Displacement of 8-hydroxy-[3H]DPAT from human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330441(3-amino-2-(4-(4-(quinolin-2-yl)piperazin-1-yl)buty...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330445(7-Acetyl-3-amino-2-[3-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330446(3-Amino-5,6-dimethyl-2-[3-(4-pyridin-2-ylpiperazin...)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330447(3-Amino-5,6-dimethyl-2-[3-[4-(4-methylquinolin-2-y...)
Affinity DataIC50:  4.30nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330448(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  5.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330440(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330449(3-Amino-5,6-dimethyl-2-[3-[4-(5,6,7,8-tetrahydroqu...)
Affinity DataIC50:  6.10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330450(2-[4-(4-Quinolin-2-ylpiperazin-1-yl)butyl]-5,6,7,8...)
Affinity DataIC50:  6.20nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330451(5-Amino-2-[5-(4-quinolin-2-ylpiperazin-1-yl)pentyl...)
Affinity DataIC50:  7.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330441(3-amino-2-(4-(4-(quinolin-2-yl)piperazin-1-yl)buty...)
Affinity DataIC50:  8.90nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330441(3-amino-2-(4-(4-(quinolin-2-yl)piperazin-1-yl)buty...)
Affinity DataIC50: >8.93nMAssay Description:Displacement of [3H]BRL-43694 from human recombinant 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330452(3-Amino-5-methyl-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  13.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330454(3-Amino-8-methyl-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  15.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330455(3-Amino-7-chloro-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330456(7-Acetyl-3-amino-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  22.1nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330457(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  24.4nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330450(2-[4-(4-Quinolin-2-ylpiperazin-1-yl)butyl]-5,6,7,8...)
Affinity DataIC50:  24.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330458(3-Amino-5,6-dimethyl-2-[4-(4-quinolin-2-ylpiperazi...)
Affinity DataIC50:  26.7nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330460(3-Amino-5,6-dimethyl-2-[3-(4-quinolin-2-ylpiperazi...)
Affinity DataIC50:  36.4nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330461(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  41.4nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330462(2-[3-(4-Quinolin-2-ylpiperazin-1-yl)propylthio]-5,...)
Affinity DataIC50:  44.2nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330463(3-Amino-6-methyl-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  45.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330459(3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]...)
Affinity DataIC50:  45.7nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330464(3-Amino-6-hydroxy-2-[4-(4-quinolin-2-ylpiperazin-1...)
Affinity DataIC50:  46.5nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330465(3-Amino-2-[4-[4-(7-hydroxyquinolin-2-yl)piperazin-...)
Affinity DataIC50:  46.6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330466(3-Amino-6-methyl-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  48.3nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330460(3-Amino-5,6-dimethyl-2-[3-(4-quinolin-2-ylpiperazi...)
Affinity DataIC50:  48.4nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330447(3-Amino-5,6-dimethyl-2-[3-[4-(4-methylquinolin-2-y...)
Affinity DataIC50:  50.5nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330467(3-Amino-5-fluoro-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  50.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330443(3-Amino-2-[4-[4-(3-hydroxyquinolin-2-yl)piperazin-...)
Affinity DataIC50:  52.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330465(3-Amino-2-[4-[4-(7-hydroxyquinolin-2-yl)piperazin-...)
Affinity DataIC50:  55.2nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330468(3-Amino-5,6-dimethyl-2-[3-(4-phenanthridin-6-ylpip...)
Affinity DataIC50:  55.4nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330453(3-Amino-2-[4-[4-(4-methylquinolin-2-yl)piperazin-1...)
Affinity DataIC50:  59.1nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330471(3-Amino-2-[4-[4-(6-hydroxyquinolin-2-yl)piperazin-...)
Affinity DataIC50:  59.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330472(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  61nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330473(3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]...)
Affinity DataIC50:  62.1nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330474(3-Amino-2-[4-[4-(2,3-dihydro-1H-cyclopenta[c]quino...)
Affinity DataIC50:  62.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330440(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  63.8nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330475(3-Amino-2-[4-[4-(3,4-dimethylquinolin-2-yl)piperaz...)
Affinity DataIC50:  64.6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330476(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  64.8nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330477(3-Amino-2-[3-(4-benzothiazol-2-ylpiperazin-1-yl)pr...)
Affinity DataIC50:  66.6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330457(3-Amino-2-[3-(4-quinolin-2-ylpiperazin-1-yl)propyl...)
Affinity DataIC50:  69.9nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330445(7-Acetyl-3-amino-2-[3-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  77.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330478(3-Amino-8-chloro-2-[4-(4-quinolin-2-ylpiperazin-1-...)
Affinity DataIC50:  83.1nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330479(3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]...)
Affinity DataIC50:  84.8nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330480(3-Amino-2-[2-(4-quinolin-2-ylpiperazin-1-yl)methyl...)
Affinity DataIC50:  86.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A(Human)
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330477(3-Amino-2-[3-(4-benzothiazol-2-ylpiperazin-1-yl)pr...)
Affinity DataIC50:  87.6nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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