Compile Data Set for Download or QSAR
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Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50032490
TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39156(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...)
Affinity DataIC50:  240nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313364((2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphen...)
Affinity DataIC50:  250nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39146(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...)
Affinity DataIC50:  300nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39124(3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...)
Affinity DataIC50:  300nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39146(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...)
Affinity DataIC50:  400nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39124(3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...)
Affinity DataIC50:  400nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313335(6-(cyclohexylamino)-N-(4-sulfamoylphenyl)pyrimidin...)
Affinity DataIC50:  450nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM34194(3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-methylpipe...)
Affinity DataIC50:  600nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39147(3-chloranyl-1-(3,4-dichlorophenyl)-4-[(3R)-3-methy...)
Affinity DataIC50:  600nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39156(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...)
Affinity DataIC50:  620nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39149(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[(E)-3-phe...)
Affinity DataIC50:  690nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313335(6-(cyclohexylamino)-N-(4-sulfamoylphenyl)pyrimidin...)
Affinity DataIC50:  800nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39147(3-chloranyl-1-(3,4-dichlorophenyl)-4-[(3R)-3-methy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM34194(3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-methylpipe...)
Affinity DataIC50:  800nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313365((2R,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylbenz...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39143(3-chloranyl-1-(2-chlorophenyl)-4-(4-methylpiperazi...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313363(3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39144(3-chloranyl-1-(3-chlorophenyl)-4-(4-methylpiperazi...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39162(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(3-methoxy...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39152(3-(4-benzylpiperazin-1-yl)-4-chloro-1-(3,4-dichlor...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313354(6-((cyclopropylmethyl)(propyl)amino)-N-(6-methyl-1...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313365((2R,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylbenz...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313353(6-(cyclohexyl(cyclopropylmethyl)amino)-N-(6-methyl...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39164(3-chloranyl-1-(3,4-dichlorophenyl)-4-(2-methyl-3-o...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39144(3-chloranyl-1-(3-chlorophenyl)-4-(4-methylpiperazi...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313366((2R,3S,4R,6R)-6-(3-(4-ethylbenzyl)-4-methylphenyl)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313363(3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313353(6-(cyclohexyl(cyclopropylmethyl)amino)-N-(6-methyl...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39152(3-(4-benzylpiperazin-1-yl)-4-chloro-1-(3,4-dichlor...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39141(1-[2,3-bis(chloranyl)phenyl]-3-chloranyl-4-(4-meth...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313354(6-((cyclopropylmethyl)(propyl)amino)-N-(6-methyl-1...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39160(3-(4-butyl-1-piperazinyl)-4-chloro-1-(3,4-dichloro...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39143(3-chloranyl-1-(2-chlorophenyl)-4-(4-methylpiperazi...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39176(3-chloranyl-4-(4-methylpiperazin-1-yl)-1-(3-nitrop...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39154(3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-phenylpipe...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313366((2R,3S,4R,6R)-6-(3-(4-ethylbenzyl)-4-methylphenyl)...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313369((6S,7R,8R,9S)-6-(4-chloro-3-(4-methoxybenzyl)pheny...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39162(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(3-methoxy...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39164(3-chloranyl-1-(3,4-dichlorophenyl)-4-(2-methyl-3-o...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39157(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-methoxy...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39176(3-chloranyl-4-(4-methylpiperazin-1-yl)-1-(3-nitrop...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39159(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(4-methoxy...)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39141(1-[2,3-bis(chloranyl)phenyl]-3-chloranyl-4-(4-meth...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM39157(3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-methoxy...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50330073(1-(3,4-dichlorophenyl)-3-(4-methylpiperazin-1-yl)p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50330072(1-(4-chlorophenyl)-3-(4-methylpiperazin-1-yl)-1H-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50330070(3-chloro-1-(3,4-dichlorophenyl)-4-(4-(3-trifluorom...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50330069(3-chloro-1-(3,4-dichlorophenyl)-4-(4-(3-methylphen...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50330073(1-(3,4-dichlorophenyl)-3-(4-methylpiperazin-1-yl)p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBcl-2-related protein A1(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50313374((5S,6R,7R,8S)-5-(3-(4-ethylbenzyl)-4-methylphenyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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