Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50032532
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330657BDBM50330657(2-(4-tert-Butylbenzyl)-3-[2-(4-hydroxy-3-iodo-5-me...)
Affinity DataKi:  2.80nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330677BDBM50330677(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-bromo-5-met...)
Affinity DataKi:  3.40nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330680BDBM50330680(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3,5-dichlorop...)
Affinity DataKi:  3.96nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330654BDBM50330654(N-[3-pivaloyloxy-2-(4-t-butylbenzyl)propyl]-2-(4-h...)
Affinity DataEC50:  4.08nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as increase of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330676BDBM50330676(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-chloro-5-me...)
Affinity DataKi:  4.09nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330672BDBM50330672(2-(4-tert-Butylbenzyl)-3-[2-(3,5-dichloro-4-hydrox...)
Affinity DataKi:  4.26nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330681BDBM50330681(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3,5-dibromoph...)
Affinity DataKi:  4.30nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330656BDBM50330656(2-(4-tert-Butylbenzyl)-3-[2-(3-bromo-4-hydroxy-5-m...)
Affinity DataKi:  8.77nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330672BDBM50330672(2-(4-tert-Butylbenzyl)-3-[2-(3,5-dichloro-4-hydrox...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330656BDBM50330656(2-(4-tert-Butylbenzyl)-3-[2-(3-bromo-4-hydroxy-5-m...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330680BDBM50330680(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3,5-dichlorop...)
Affinity DataKi:  9.43nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330673BDBM50330673(2-(4-tert-Butylbenzyl)-3-[2-(3,5-dibromo-4-hydroxy...)
Affinity DataKi:  10.7nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330681BDBM50330681(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3,5-dibromoph...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330654BDBM50330654(N-[3-pivaloyloxy-2-(4-t-butylbenzyl)propyl]-2-(4-h...)
Affinity DataKi:  13.1nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330660BDBM50330660(2-(4-tert-Butylbenzyl)-3-[2-(4-hydroxy-2-iodo-5-me...)
Affinity DataKi:  13.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330662BDBM50330662(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-3-bromo-5-m...)
Affinity DataKi:  13.6nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330644BDBM50330644(N-(4-tert-Butyl-benzyl)-2-(3-iodo-4-hydroxy-5-meth...)
Affinity DataKi:  17.2nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330663BDBM50330663(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-3-iodo-5-me...)
Affinity DataKi:  19.1nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330666BDBM50330666(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-2-iodo-5-me...)
Affinity DataKi:  19.5nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330673BDBM50330673(2-(4-tert-Butylbenzyl)-3-[2-(3,5-dibromo-4-hydroxy...)
Affinity DataKi:  20.2nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330663BDBM50330663(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-3-iodo-5-me...)
Affinity DataKi:  20.3nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330660BDBM50330660(2-(4-tert-Butylbenzyl)-3-[2-(4-hydroxy-2-iodo-5-me...)
Affinity DataKi:  20.9nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330661BDBM50330661(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-3-chloro-5-...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330657BDBM50330657(2-(4-tert-Butylbenzyl)-3-[2-(4-hydroxy-3-iodo-5-me...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330675BDBM50330675(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-methoxyphen...)
Affinity DataEC50:  22.9nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as increase of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330664BDBM50330664(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-2-chloro-5-...)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330671BDBM50330671(3-[2-(3-Bromo-4-hydroxyphenyl)acetamido]-2-(4-tert...)
Affinity DataKi:  25.1nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330659BDBM50330659(2-(4-tert-Butylbenzyl)-3-[2-(2-bromo-4-hydroxy-5-m...)
Affinity DataKi:  25.3nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330655BDBM50330655(2-(4-tert-Butylbenzyl)-3-[2-(3-chloro-4-hydroxy-5-...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330676BDBM50330676(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-chloro-5-me...)
Affinity DataKi:  33.5nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330665BDBM50330665(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-2-bromo-5-m...)
Affinity DataKi:  34.9nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330658BDBM50330658(2-(4-tert-Butylbenzyl)-3-[2-(2-chloro-4-hydroxy-5-...)
Affinity DataKi:  37.6nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330683BDBM50330683(2-(4-tert-Butylbenzyl)-3-[2-(2-bromo-4-methanesulf...)
Affinity DataKi:  42.9nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330650BDBM50330650(N-(4-tert-Butyl-benzyl)-2-(4-acetoxy-3-iodo-5-meth...)
Affinity DataKi:  47.9nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330666BDBM50330666(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-2-iodo-5-me...)
Affinity DataKi:  53nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330667BDBM50330667(3-[2-(3-Bromo-4-hydroxy-5-methoxyphenyl)acetamido]...)
Affinity DataKi:  56.4nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330679BDBM50330679(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-bromophenyl...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330662BDBM50330662(2-(4-tert-Butylbenzyl)-3-[2-(4-acetoxy-3-bromo-5-m...)
Affinity DataKi:  72nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330677BDBM50330677(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-bromo-5-met...)
Affinity DataKi:  79.1nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330641BDBM50330641(N-(4-t-butylbenzyl)-2-(4-hydroxy-3-methoxyphenyl)a...)
Affinity DataEC50:  82nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as increase of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330682BDBM50330682(2-(4-tert-Butylbenzyl)-3-[2-(4-methanesulfonylamin...)
Affinity DataKi:  84.5nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330644BDBM50330644(N-(4-tert-Butyl-benzyl)-2-(3-iodo-4-hydroxy-5-meth...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330643BDBM50330643(N-(4-tert-Butyl-benzyl)-2-(3-bromo-4-hydroxy-5-met...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330650BDBM50330650(N-(4-tert-Butyl-benzyl)-2-(4-acetoxy-3-iodo-5-meth...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330674BDBM50330674(2-(4-tert-Butylbenzyl)-3-[2-(3,5-dibromophenyl)ace...)
Affinity DataKi:  108nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330675BDBM50330675(2-(4-tert-Butylbenzyl)-3-[2-(4-amino-3-methoxyphen...)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330670BDBM50330670(2-(3,4-Dimethylbenzyl)-3-[2-(4-hydroxy-2-iodo-5-me...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170053BDBM50170053(N-(4-hydroxy-2-iodo-5-methoxybenzyl)nonanamide | N...)
Affinity DataKi:  127nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330645BDBM50330645(N-(4-tert-Butyl-benzyl)-2-(2-chloro-4-hydroxy-5-me...)
Affinity DataEC50:  135nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as increase of capsaicin-induced calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330642BDBM50330642(N-(4-tert-Butyl-benzyl)-2-(3-chloro-4-hydroxy-5-me...)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
Displayed 1 to 50 (of 67 total ) | Next | Last >>
Jump to: