Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50032578
LigandPNGBDBM50331363((S)-3'-cyclopropyl-4'-(4-(1,1,1-trifluoro-2-hydrox...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50248569((1-(((R)-3-methyl-4-(4-((S)-1,1,1-trifluoro-2-hydr...)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331361((S)-3'-chloro-4'-(4-(1,1,1-trifluoro-2-hydroxyprop...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331341(rac-2-(4-(2-ethylphenylsulfonyl)phenyl)-1,1,1-trif...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331343(rac-2-(4-(2-cyclopropylphenylsulfonyl)phenyl)-1,1,...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331365((S)-3'-(2-fluoroethyl)-4'-(4-(1,1,1-trifluoro-2-hy...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331350(rac-2-(4-(4-bromo-2-chlorophenylsulfonyl)phenyl)-1...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331349(rac-2-(4-(2,4-dichlorophenylsulfonyl)phenyl)-1,1,1...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331363((S)-3'-cyclopropyl-4'-(4-(1,1,1-trifluoro-2-hydrox...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331351(rac-3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypropan...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331352(rac-2-(4-(2-chloro-4-nitrophenylsulfonyl)phenyl)-1...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331342(rac-1,1,1-trifluoro-2-(4-(2-isopropylphenylsulfony...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331330(rac-1,1,1-trifluoro-2-(4-(o-tolylsulfonyl)phenyl)p...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331329(rac-2-(4-(2-chlorophenylsulfonyl)phenyl)-1,1,1-tri...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331354(rac-2-(4-(2-chloro-4-(pyridin-4-yl)phenylsulfonyl)...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50248569((1-(((R)-3-methyl-4-(4-((S)-1,1,1-trifluoro-2-hydr...)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331340(rac-1,1,1-trifluoro-2-(4-(2-(trifluoromethyl)pheny...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331358(rac-1-(3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypro...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331344(rac-2-(4-(2-tert-butylphenylsulfonyl)phenyl)-1,1,1...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331339(rac-1,1,1-trifluoro-2-(4-(2-fluorophenylsulfonyl)p...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331361((S)-3'-chloro-4'-(4-(1,1,1-trifluoro-2-hydroxyprop...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331362((R)-3'-cyclopropyl-4'-(4-(1,1,1-trifluoro-2-hydrox...)
Affinity DataIC50: 11.2nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331360((R)-3'-chloro-4'-(4-(1,1,1-trifluoro-2-hydroxyprop...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331356(rac-3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypropan...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331331(rac-2-(4-(3-chlorophenylsulfonyl)phenyl)-1,1,1-tri...)
Affinity DataIC50: 18.1nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331337(rac-1-(4-tert-butylphenylsulfonyl)-2-chlorobenzene...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331365((S)-3'-(2-fluoroethyl)-4'-(4-(1,1,1-trifluoro-2-hy...)
Affinity DataIC50: 20.7nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331353(rac-3'-chloro-4'-(4-(1,1,1-trifluoro-2-hydroxyprop...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331334(rac-1,1,1-trifluoro-2-(4-(4-nitrophenylsulfonyl)ph...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331343(rac-2-(4-(2-cyclopropylphenylsulfonyl)phenyl)-1,1,...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331332(rac-1,1,1-trifluoro-2-(4-(4-methoxyphenylsulfonyl)...)
Affinity DataIC50: 28.7nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331359(rac-1-(3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypro...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331355(rac-2-(4-(4-amino-2-chlorophenylsulfonyl)phenyl)-1...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331336(rac-1-chloro-2-(4-(2-fluoropropan-2-yl)phenylsulfo...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331364((R)-3'-(2-fluoroethyl)-4'-(4-(1,1,1-trifluoro-2-hy...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331333(rac-1,1,1-trifluoro-2-(4-(4-fluorophenylsulfonyl)p...)
Affinity DataIC50: 36.6nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331351(rac-3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypropan...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331349(rac-2-(4-(2,4-dichlorophenylsulfonyl)phenyl)-1,1,1...)
Affinity DataIC50: 43nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331329(rac-2-(4-(2-chlorophenylsulfonyl)phenyl)-1,1,1-tri...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331345(rac-2-(4-(1,1,1-trifluoro-2-hydroxypropan-2-yl)phe...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331330(rac-1,1,1-trifluoro-2-(4-(o-tolylsulfonyl)phenyl)p...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331350(rac-2-(4-(4-bromo-2-chlorophenylsulfonyl)phenyl)-1...)
Affinity DataIC50: 59nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331328(rac-1,1,1-trifluoro-2-(4-(phenylsulfonyl)phenyl)pr...)
Affinity DataIC50: 79nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331357(rac-1-(3-chloro-4-(4-(1,1,1-trifluoro-2-hydroxypro...)
Affinity DataIC50: 86nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331341(rac-2-(4-(2-ethylphenylsulfonyl)phenyl)-1,1,1-trif...)
Affinity DataIC50: 93nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331335(rac-2-(4-(2-chlorophenylsulfonyl)phenyl)propan-2-o...)
Affinity DataIC50: 102nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331352(rac-2-(4-(2-chloro-4-nitrophenylsulfonyl)phenyl)-1...)
Affinity DataIC50: 105nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331346(rac-1,1,1-trifluoro-2-(4-(4'-fluorobiphenyl-2-ylsu...)
Affinity DataIC50: 109nMAssay Description:Inhibition of human 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331354(rac-2-(4-(2-chloro-4-(pyridin-4-yl)phenylsulfonyl)...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50331362((R)-3'-cyclopropyl-4'-(4-(1,1,1-trifluoro-2-hydrox...)
Affinity DataIC50: 125nMAssay Description:Inhibition of human 11beta-HSD1 transfected in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
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