TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Binding affinity to human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Binding affinity to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 13.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 22.6nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Displacement of [3H]SCH 23990 from dopamine D1 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]SCH 23990 from dopamine D1 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataEC50: 3.90nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO dhfr-negative cells assessed as stimulation of [3H]-thymidine incorporationMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at human dopamine receptor D2long expressed in CHO10001 cells assessed as stimulation of incorporation [3H]-thymidine incorporationMore data for this Ligand-Target Pair