Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50032734
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333919BDBM50333919((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324822BDBM50324822((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 5nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333915BDBM50333915((S)-2-(2-(benzofuran-2-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 5nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333917BDBM50333917((S)-2-(5,7-dichloro-2-(pyrazolo[1,5-a]pyridine-2-c...)
Affinity DataIC50: 7nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333916BDBM50333916((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 19nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324812BDBM50324812((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 22nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333904BDBM50333904((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 26nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333918BDBM50333918((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 30nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333905BDBM50333905((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 39nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333911BDBM50333911((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 59nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333919BDBM50333919((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 96nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333901BDBM50333901((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 100nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333906BDBM50333906((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 140nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333921BDBM50333921((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 150nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333909BDBM50333909((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 170nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333915BDBM50333915((S)-2-(2-(benzofuran-2-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 190nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333913BDBM50333913((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 250nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333917BDBM50333917((S)-2-(5,7-dichloro-2-(pyrazolo[1,5-a]pyridine-2-c...)
Affinity DataIC50: 260nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333912BDBM50333912((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 310nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333907BDBM50333907((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 430nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333908BDBM50333908((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 560nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333918BDBM50333918((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 560nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50125195BDBM50125195((S)-2-(2-Bromo-benzoylamino)-3-(3H-imidazol-4-yl)-...)
Affinity DataIC50: 750nMAssay Description:Inhibition of LFA1/ICAM1 interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333899BDBM50333899((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 810nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333900BDBM50333900((S)-3-(1-acetyl-1H-indole-3-carboxamido)-2-(5,7-di...)
Affinity DataIC50: 820nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333916BDBM50333916((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 950nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324822BDBM50324822((S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2,...)
Affinity DataIC50: 950nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333920BDBM50333920((S)-ethyl 2-(2-(benzofuran-6-carbonyl)-5,7-dichlor...)
Affinity DataIC50: 950nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333911BDBM50333911((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333902BDBM50333902((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333922BDBM50333922((2S)-2-(2-(benzofuran-6-carbonyl)-5,7-dichloro-1,2...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333903BDBM50333903((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333914BDBM50333914((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333910BDBM50333910((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50324812BDBM50324812((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50125228BDBM50125228((S)-2-(2-Bromo-benzoylamino)-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of LFA1/ICAM1 interaction by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333904BDBM50333904((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333906BDBM50333906((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333901BDBM50333901((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetIntegrin alpha-L/beta-2(Human)
Sunesis Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333905BDBM50333905((S)-2-(5,7-dichloro-2-(4-chlorobenzoyl)-1,2,3,4-te...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of LFA1/ICAM1 interaction in human Hut-78 cells in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed