Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 5718
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341682(6,6'-(2,2'-(Pyridine-3,5-diyl)bis(ethane-2,1-diyl)...)
Affinity DataKi:  25nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341684(6,6'-(2,2'-(1,3-Phenylene)bis(ethane-2,1-diyl))bis...)
Affinity DataKi:  38nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341678(6,6'-(2,2'-(5-Amino-1,3-phenylene)bis(ethane-2,1di...)
Affinity DataKi:  85nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341681(4-(2-(5-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  103nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341679(4-(2-(6-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  195nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341682(6,6'-(2,2'-(Pyridine-3,5-diyl)bis(ethane-2,1-diyl)...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341681(4-(2-(5-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  1.91E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341682(6,6'-(2,2'-(Pyridine-3,5-diyl)bis(ethane-2,1-diyl)...)
Affinity DataKi:  2.68E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341684(6,6'-(2,2'-(1,3-Phenylene)bis(ethane-2,1-diyl))bis...)
Affinity DataKi:  2.73E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341678(6,6'-(2,2'-(5-Amino-1,3-phenylene)bis(ethane-2,1di...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341684(6,6'-(2,2'-(1,3-Phenylene)bis(ethane-2,1-diyl))bis...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341680(6,6'-(2,2'-(Pyridine-2,6-diyl)bis(ethane-2,1-diyl)...)
Affinity DataKi:  4.75E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341678(6,6'-(2,2'-(5-Amino-1,3-phenylene)bis(ethane-2,1di...)
Affinity DataKi:  4.95E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341680(6,6'-(2,2'-(Pyridine-2,6-diyl)bis(ethane-2,1-diyl)...)
Affinity DataKi:  9.40E+3nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341679(4-(2-(6-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  1.26E+4nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341681(4-(2-(5-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  1.61E+4nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University of California Irvine

LigandPNGBDBM50341679(4-(2-(6-(2-(6-Amino-4-methylpyridin-2-yl)ethyl)pyr...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition assay using nitric oxide synthases.More data for this Ligand-Target Pair