Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50032973
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337153(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  13nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337152(CHEMBL1682747 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  15nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334829(CHEMBL1643161 | N-(4-(5-cyano-7-methylbenzo[d]oxaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337194(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  19nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337173(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  22nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337189(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  22nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337188(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  24nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337190(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  28nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337192(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  29nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337193(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  31nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337175(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  37nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337186(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  39nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337172(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  40nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337184(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  43nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337187(CHEMBL1684864 | N-((1-(5-(2-chloro-6-methoxyphenyl...)
Affinity DataIC50:  47nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337185(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  48nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337177(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  61nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337176(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  110nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337174(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  114nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337178(CHEMBL1684855 | methyl 6-(4-((4-(5-cyano-7-isoprop...)
Affinity DataIC50:  114nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337171(4-(5-cyano-7-(prop-1-en-2-yl)benzo[d]oxazol-2-yl)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337170(4-(7-tert-butyl-5-cyanobenzo[d]oxazol-2-yl)-N-((1-...)
Affinity DataIC50:  198nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337182(CHEMBL1684859 | N-((1-(5-bromopyridin-2-yl)piperid...)
Affinity DataIC50:  223nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337183(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50:  229nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337168(4-(5-cyano-7-cyclopropylbenzo[d]oxazol-2-yl)-N-((1...)
Affinity DataIC50:  243nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337166(4-(5-cyano-7-methylbenzo[d]oxazol-2-yl)-N-((1-(4-(...)
Affinity DataIC50:  300nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337179(CHEMBL1684856 | methyl 6-(4-((4-(5-cyano-7-isoprop...)
Affinity DataIC50:  306nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337191(CHEMBL1684868 | N-((1-(5-(2-(benzyloxy)-5-(trifluo...)
Affinity DataIC50:  413nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337161(2-(4-(2-hydroxy-3-(4-(4-(trifluoromethyl)phenyl)pi...)
Affinity DataIC50:  874nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337154(7-methyl-2-(4-(3-(4-(4-(trifluoromethyl)phenyl)pip...)
Affinity DataIC50:  975nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337156(7-methyl-2-(4-(3-(4-(4-(trifluoromethyl)phenyl)pip...)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337155(7-methyl-2-(4-(3-(4-(4-(trifluoromethyl)phenyl)pip...)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337160(2-(4-(1-hydroxy-3-(4-(4-(trifluoromethyl)phenyl)pi...)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337167(4-(5-cyano-7-methylbenzo[d]oxazol-2-yl)-N-methyl-N...)
Affinity DataIC50:  2.61E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337164(7-methyl-2-(4-(2-oxo-3-(4-(4-(trifluoromethyl)phen...)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337169(4-(5-cyano-7-(trifluoromethyl)benzo[d]oxazol-2-yl)...)
Affinity DataIC50:  3.19E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337158(7-methyl-2-(4-(4-(4-(trifluoromethyl)phenyl)pipera...)
Affinity DataIC50:  4.03E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337159(7-methyl-2-(4-((4-(4-(trifluoromethyl)phenyl)piper...)
Affinity DataIC50:  4.55E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337157(7-methyl-2-(4-(2-oxo-3-(4-(4-(trifluoromethyl)phen...)
Affinity DataIC50:  5.74E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337162(2-(4-(2-methoxy-3-(4-(4-(trifluoromethyl)phenyl)pi...)
Affinity DataIC50:  8.94E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337181(4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)-N-((1-(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337180(6-(4-((4-(5-cyano-7-isopropylbenzo[d]oxazol-2-yl)b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337165(4-(5-cyano-7-methylbenzo[d]oxazol-2-yl)-N-(2-(1-(4...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50337163(2-(4-(2-hydroxy-3-(4-(4-(trifluoromethyl)phenyl)pi...)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed