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Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50032693
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed