Compile Data Set for Download or QSAR
maximum 50k data
Found 83 Enz. Inhib. hit(s) with all data for entry = 50032859
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335797(2-[2-(3-(R)-Aminopyrimidin-1-yl)-5-bromo-6-oxo-6H-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335792(2-{6-[3(R)-Aminopiperidin-1-yl]-2,4-dioxo-3,4-dihy...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335768(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-methoxy-6-oxo-6...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335784(2-[6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335774(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-bromo-6-oxopyr...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335756(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-prop-1-ynyl-6-o...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335757(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-ethynyl-6-oxo-6...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335759(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-5-(1H-pyrro...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335798(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-5-((E)-2-py...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335777(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-fluoro-6-oxo-6H...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335793(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-bromo-6-oxopyr...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335771(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-iodo-6-oxo-6H-p...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335775(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-chloro-6-oxo-6H...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335773(2[2-(3-(R)-Aminopiperidin-1-yl)-5-bromo-4-methyl-6...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335753(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-5-vinyl-6H-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335787(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-bromo-5-fluorob...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335795(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-fluoro-6-oxopy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335794(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-chloro-6-oxopy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335778(2-((6-(3-(R)-Amino-3-methylpiperidin-1-yl)-3-methy...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335770(2-[2-(3-(R)-Aminopiperidin-1-yl)-4,5-dimethyl-6-ox...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335761(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-furan-3-yl-6-ox...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335788(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-bromobenzyl)-3-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335766((R)-2-{[2-(3-Aminopiperidin-1-yl)-4-oxo-5,6,7,8-te...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335776(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-6H-pyrimidi...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335786(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-chloro-5-fluoro...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335769(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-ethyl-6-oxo-6H-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335755(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-(3-hydroxyprop-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335799(2-{2-(3-(R)-Aminopiperidin-1-yl)-5-[2-trans-(4-flu...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335800(2-[2-(3-(R)-Aminopiperidin-1-yl)-4-methyl-6-oxo-5-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335765(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-5-phenyl-6H...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335767(2-[2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-4-phenyl-6H...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335783(6-[3-(R)-Aminopiperidin-1-yl]-1-(2,5-dichlorobenzy...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335789(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-bromobenzyl)-1H...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335791(2-{6-[3(R)-Aminopiperidin-1-yl]-5-chloro-3-methyl-...)
Affinity DataIC50:  57nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335790(2-{6-[3(R)-Aminopiperidin-1-yl]-3-ethyl-2,4-dioxo-...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335760(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-furan-3-yl-4-me...)
Affinity DataIC50:  77nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335758(2-((2-(3-(R)-Aminopiperidin-1-yl)-6-oxo-5-(pyrroli...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335763(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-(2-fluorophenyl...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335796(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-fluoro-6-oxopy...)
Affinity DataIC50:  430nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335764(2-[2-(3-(R)-Aminopiperidin-1-yl)-4-methyl-6-oxo-5-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335754(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-(3,3-dimethylbu...)
Affinity DataIC50:  570nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335780((+/-)-2-{6-[Azepan-3((+/-)-ylamino]-3-methyl-2,4-d...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335782(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-chloro-3,6-difl...)
Affinity DataIC50:  830nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335785(6-[3-(R)-Aminopiperidin-1-yl]-1-(2-chloro-4-fluoro...)
Affinity DataIC50:  890nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335762(2-[2-(3-(R)-Aminopiperidin-1-yl)-5-(2-methoxypheny...)
Affinity DataIC50:  990nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335779((+/-)2-{6-[3((+/-)-Aminoazepan-1-yl]-3-methyl-2,4-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335772(2-((2-(3-(R)-Aminopiperidin-1-yl)-5-bromo-4-tert-b...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335781(2-[6-(2-Aminoethylamino)-3-ethyl-2,4-dioxo-3,4-dih...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50335799(2-{2-(3-(R)-Aminopiperidin-1-yl)-5-[2-trans-(4-flu...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human DPP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 83 total ) | Next | Last >>
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