Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50032717
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333656BDBM50333656((2,3-dichlorophenyl)(4-(3-(thiazol-2-ylamino)benzy...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 14192BDBM14192(3-({7-cyclohexyl-7H-pyrrolo[2,3-d]pyrimidin-2-yl}a...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13534BDBM13534(VX680 | N-[4-[[4-(4-methylpiperazino)-6-[(5-methyl...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333657BDBM50333657((4-((6-(1H-pyrazol-3-ylamino)pyridin-2-yl)methyl)p...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12103BDBM12103(CHEMBL484007 | 4-tert-butyl-N-[5-(thien-2-ylacetyl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333658BDBM50333658(N-(4-(3-(3-amino-1H-pyrazol-4-yl)pyridin-2-yloxy)p...)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333666BDBM50333666(N-(1-(2,4-dimethylphenylamino)-3-(4-hydroxyphenyl)...)
Affinity DataIC50: 5.09E+3nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333664BDBM50333664(2-amino-N-(3-(4-hydroxyphenyl)-1-oxo-1-(p-tolylami...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333663BDBM50333663(2-(6-ethoxy-4-methylquinazolin-2-ylamino)quinazoli...)
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333662BDBM50333662(7-(2-hydroxy-3-(4-methoxyphenoxy)propyl)-8-(2-(2-h...)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333661BDBM50333661(N-(2-cyclohexenylethyl)-2-(4-(6-methoxy-1H-indole-...)
Affinity DataIC50: 8.62E+4nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333665BDBM50333665(N-(4-ethoxyphenyl)-2-(8-(4-ethoxyphenylamino)-3-me...)
Affinity DataIC50: 9.87E+4nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333659BDBM50333659(6-(3,4-dimethoxyphenyl)-N-(2,4-dimethylphenyl)-3-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333660BDBM50333660(N1-(3-acetamidophenyl)-N2-(2-(2-(4-chlorophenyl)-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50333667BDBM50333667(N-(5-bromothiazol-2-yl)-2-(5-methoxybenzo[d]thiazo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant His-tagged Aurora A kinase expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed