Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 163 Enz. Inhib. hit(s) with all data for entry = 50039378
TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268876(CHEMBL509572 | Disodium 1-amino-4-[4-(4-chloro-6-m...)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50029031(1-Amino-4-{4-[4-chloro-6-(3-sulfo-phenylamino)-[1,...)
Affinity DataKi:  680nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268874(CHEMBL499580 | Sodium 1-Amino-4-[3-(4,6-dichloro-[...)
Affinity DataKi:  3.76E+3nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227020(CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylami...)
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227032(CHEMBL256057 | acid blue 25 | sodium 1-amino-9,10-...)
Affinity DataKi:  9.83E+3nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336787(CHEMBL445413 | sodium 1-amino-9,10-dioxo-4-(m-toly...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336768(CHEMBL1671995 | sodium 1-amino-4-(3-methoxyphenyla...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2Y purinoceptor 12(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataKi:  1.71E+4nMAssay Description:Displacement of [3H]PSB0413 from human platelet P2Y12 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataIC50:  79nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336796(CHEMBL1672105 | Sodium 1-Amino-4-[3-(4,6-dichloro[...)
Affinity DataIC50:  86nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227020(CHEMBL271672 | sodium 1-amino-4-(3-chlorophenylami...)
Affinity DataIC50:  100nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268875(CHEMBL496401 | Sodium 1-amino-4-[4-(4,6-dichloro-[...)
Affinity DataIC50:  117nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336782(CHEMBL1672106 | Sodium 1-Amino-4-[4-(4,6-dihydroxy...)
Affinity DataIC50:  197nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268874(CHEMBL499580 | Sodium 1-Amino-4-[3-(4,6-dichloro-[...)
Affinity DataIC50:  293nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336797(CHEMBL1672107 | Disodium 1-Amino-4-[3-(4,6-dihydro...)
Affinity DataIC50:  300nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 1(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataIC50:  422nMAssay Description:Antagonist activity against rat P2X1 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 3(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336781(CHEMBL1672104 | Disodium 1-Amino-4-[3-(4,6-dichlor...)
Affinity DataIC50:  494nMAssay Description:Antagonist activity against rat P2X3 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268876(CHEMBL509572 | Disodium 1-amino-4-[4-(4-chloro-6-m...)
Affinity DataIC50:  582nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268725(CHEMBL496030 | sodium 1-amino-4-(4-hydroxyphenylam...)
Affinity DataIC50:  588nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336768(CHEMBL1671995 | sodium 1-amino-4-(3-methoxyphenyla...)
Affinity DataIC50:  623nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227015(CHEMBL271688 | Sodium 1-amino-4-(4-acetylaminophen...)
Affinity DataIC50:  690nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336787(CHEMBL445413 | sodium 1-amino-9,10-dioxo-4-(m-toly...)
Affinity DataIC50:  800nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336772(CHEMBL1672098 | sodium 1-amino-4-(3-bromophenylami...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50118231(CHEMBL134193 | Cibachron Blue 3GA)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268686(CHEMBL496022 | sodium 1-amino-9,10-dioxo-4-(4-sulf...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268685(CHEMBL524064 | sodium 1-amino-4-(2-carboxyphenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336774(CHEMBL598857 | sodium 1-amino-4-(3-carboxyphenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336775(CHEMBL604300 | sodium 1-amino-4-(4-carboxyphenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268635(CHEMBL450832 | sodium 1-amino-4-(2-aminophenylamin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336776(CHEMBL597820 | sodium 1-amino-4-(3-aminophenylamin...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336771(CHEMBL604158 | sodium 1-amino-4-(4-fluorophenylami...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336794(CHEMBL1671997 | Sodium 1-amino-4-(3-flourophenylam...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336770(CHEMBL597203 | Sodium 1-amino-4-(4-phenoxyphenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336769(CHEMBL403051 | sodium 1-amino-4-(2-ethoxyphenylami...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336793(CHEMBL1671996 | Sodium 1-amino-4-(3,5-dimethoxyphe...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268687(CHEMBL522725 | sodium 1-amino-4-(2-hydroxyphenylam...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336792(CHEMBL256688 | sodium 1-amino-4-(2,4-dimethylpheny...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336791(CHEMBL402239 | sodium 1-amino-4-(2,3-dimethylpheny...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336790(CHEMBL1671993 | Sodium 1-amino-4-(3-ethylphenylami...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336789(CHEMBL1671992 | Sodium 1-amino-4-(3-trifluoromethy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336788(CHEMBL404450 | sodium 1-amino-9,10-dioxo-4-(p-toly...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336786(CHEMBL256864 | sodium 1-amino-9,10-dioxo-4-(o-toly...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336785(CHEMBL606414 | sodium 1-amino-4-(cyclohexylamino)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50227032(CHEMBL256057 | acid blue 25 | sodium 1-amino-9,10-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336795(CHEMBL1672099 | Sodium 1-amino-4-(3,5-difluorophen...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268966(CHEMBL496229 | Sodium 1-Amino-4-[4-([1,3]diazine-2...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50268965(CHEMBL499428 | Disodium 1-amino-4-[4-([1,3]diazine...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetP2X purinoceptor 2(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50336780(CHEMBL1672103 | sodium 1-amino-4-(3-amino-2-methyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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