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Found 19 Enz. Inhib. hit(s) with all data for entry = 50032881
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336049(CHEMBL1669334 | N-benzyl-4-(6-(cyclopropylmethylam...)
Affinity DataIC50:  12nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336052(CHEMBL1669337 | N-cinnamyl-4-(6-(cyclopropylmethyl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336057(CHEMBL1669342 | N-(4-acetamidobenzyl)-4-(6-(cyclop...)
Affinity DataIC50:  15nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336055(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  15nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336065(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  16nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336050(CHEMBL1669335 | N-(3-chlorobenzyl)-4-(6-(cycloprop...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336051(CHEMBL1669336 | N-(4-chlorobenzyl)-4-(6-(cycloprop...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336056(4-((4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  17nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336064(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  18nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336060(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  21nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336061(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  22nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336058(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  23nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336063(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  42nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325375((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336059(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  71nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336062((S)-4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyr...)
Affinity DataIC50:  97nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336054(2-(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyri...)
Affinity DataIC50:  110nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50325369(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  200nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336053(4-(6-(cyclopropylmethylamino)imidazo[1,2-b]pyridaz...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of purified His-tagged IKKbeta after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed