Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for entry = 50032893
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336285(6-(2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-ylamino)...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336286(6-(2-(5-((4-methylpiperazin-1-yl)methyl)pyrimidin-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336287(5-(2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-ylamino)...)
Affinity DataIC50:  18nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50335963(CHEMBL1667925 | ethyl 3-(1-(hydroxyimino)-2,3-dihy...)
Affinity DataIC50:  30nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336288(2-chloro-5-(2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3...)
Affinity DataIC50:  31nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336289(3-(5-hydroxynaphthalen-2-ylamino)-N-(pyrimidin-4-y...)
Affinity DataIC50:  37.9nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336290(CHEMBL1667906 | ethyl 3-(5-hydroxynaphthalen-2-yla...)
Affinity DataIC50:  54nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336291(3-(5-hydroxynaphthalen-2-ylamino)-N-isopropylfuro[...)
Affinity DataIC50:  86.7nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336292(CHEMBL1667909 | N-(2-(dimethylamino)vinyl)-3-(5-hy...)
Affinity DataIC50:  102nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336293(CHEMBL1667923 | N-(7-chloro-3-ethyl-1H-indazol-4-y...)
Affinity DataIC50:  140nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336294(CHEMBL1667907 | ethyl 3-(6-fluoro-5-hydroxynaphtha...)
Affinity DataIC50:  142nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336295(CHEMBL1667916 | N-(7-chloro-1H-indazol-4-yl)-2-(py...)
Affinity DataIC50:  250nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336314(CHEMBL1667922 | N-(7-chloro-6-methyl-1H-indazol-4-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336296(3-(7-chloro-4-(2-(pyrimidin-2-yl)furo[2,3-c]pyridi...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336297(CHEMBL1667912 | ethyl 3-(4-chloro-3-hydroxyphenyla...)
Affinity DataIC50:  442nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336311(3-(4-chloro-3-hydroxyphenylamino)-N-(pyrimidin-2-y...)
Affinity DataIC50:  556nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336312(5-(2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-ylamino)...)
Affinity DataIC50:  820nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336313(3-(4-chloro-3-hydroxyphenylamino)-N-isopropylfuro[...)
Affinity DataIC50:  823nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336298(CHEMBL1667920 | N-(7-methyl-1H-indazol-4-yl)-2-(py...)
Affinity DataIC50:  840nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336299(CHEMBL1667902 | N-(2,4-dihydroindeno[1,2-c]pyrazol...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336300(3-(1-(hydroxyimino)isoindolin-5-ylamino)-N-isoprop...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336301(CHEMBL1667865 | N-(3-(3-aminopropyl)-7-chloro-1H-i...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336302(CHEMBL1667917 | N-(6-chloro-1H-indazol-4-yl)-2-(py...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336303(CHEMBL1667915 | N-(1H-indazol-4-yl)-2-(pyrimidin-2...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336304(CHEMBL1667921 | N-(7-fluoro-1H-indazol-4-yl)-2-(py...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336305(3-(7-chloro-1H-indazol-4-ylamino)-N-isopropylfuro[...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336306(3-(2,4-dihydroindeno[1,2-c]pyrazol-6-ylamino)-N-(2...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336307(CHEMBL1667904 | ethyl 3-(quinolin-3-ylamino)furo[2...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336308(CHEMBL1667898 | ethyl 3-(1-oxo-2,3-dihydro-1H-inde...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336309(3-(2,4-dihydroindeno[1,2-c]pyrazol-6-ylamino)-N-is...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50336310(CHEMBL1667905 | ethyl 3-(5-aminonaphthalen-2-ylami...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of pERKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed