Compile Data Set for Download or QSAR
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Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50032939
TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50304496(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336694(3-Benzo[1,3]dioxol-5-yl-4-{3-(2-(2-(2-(2-fluoroeth...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336695(3-Benzo[1,3]dioxol-5-yl-4-{3-[1-(2-{2-[2-(2-fluoro...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336697(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{4-[4-(2-...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336699(CHEMBL1672884 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336696(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{1-[2-(2-...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336698(CHEMBL1672885 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336700(3-Benzo[1,3]dioxol-5-yl-4-{3-[2-(2-{2-[2-(4-fluoro...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336697(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{4-[4-(2-...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50304496(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...)
Affinity DataKi:  240nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336699(CHEMBL1672884 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...)
Affinity DataKi:  288nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336694(3-Benzo[1,3]dioxol-5-yl-4-{3-(2-(2-(2-(2-fluoroeth...)
Affinity DataKi:  418nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336698(CHEMBL1672885 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...)
Affinity DataKi:  893nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336696(3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{1-[2-(2-...)
Affinity DataKi:  5.34E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336700(3-Benzo[1,3]dioxol-5-yl-4-{3-[2-(2-{2-[2-(4-fluoro...)
Affinity DataKi:  6.45E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Mouse)
University Hospital Mu£Nster

Curated by ChEMBL
LigandPNGBDBM50336695(3-Benzo[1,3]dioxol-5-yl-4-{3-[1-(2-{2-[2-(2-fluoro...)
Affinity DataKi:  8.45E+3nMAssay Description:Displacement of [125I]ET1 from ETB receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed