Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50032979
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337291BDBM50337291(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337299BDBM50337299(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337301BDBM50337301(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337302BDBM50337302(3-((3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihy...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337295BDBM50337295(1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337292BDBM50337292(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337293BDBM50337293(1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337294BDBM50337294(1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337300BDBM50337300(1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337296BDBM50337296(1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337303BDBM50337303(1-(4-tert-butylbenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337298BDBM50337298(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50318159BDBM50318159(CHEMBL1095777 | 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337297BDBM50337297(1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig tracheal rings assessed as vasorelaxationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337297BDBM50337297(1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  296nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337292BDBM50337292(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  550nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337300BDBM50337300(1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337294BDBM50337294(1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50318159BDBM50318159(CHEMBL1095777 | 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-...)
Affinity DataEC50:  2.31E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337296BDBM50337296(1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...)
Affinity DataEC50:  5.77E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337293BDBM50337293(1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337295BDBM50337295(1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...)
Affinity DataEC50:  8.89E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337291BDBM50337291(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337301BDBM50337301(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337299BDBM50337299(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337298BDBM50337298(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed