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Found 48 Enz. Inhib. hit(s) with all data for entry = 50032909
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM10868(1,3,4-Thiadiazole-2-sulfonamide, 6 | 1,3,4-thiadia...)
Affinity DataKi:  33nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM10868(1,3,4-Thiadiazole-2-sulfonamide, 6 | 1,3,4-thiadia...)
Affinity DataKi:  41nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM10868(1,3,4-Thiadiazole-2-sulfonamide, 6 | 1,3,4-thiadia...)
Affinity DataKi:  60nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50100861(3,4-Dihydroxybenzoate, VIII | 3,4-dihydroxybenzoic...)
Affinity DataKi:  470nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336488(1,2-dimethoxybenzene | CHEMBL1668603)
Affinity DataKi:  500nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataKi:  510nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataKi:  550nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataKi:  600nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336492(2,6-dimethoxybenzoic acid | CHEMBL488609)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50100861(3,4-Dihydroxybenzoate, VIII | 3,4-dihydroxybenzoic...)
Affinity DataKi:  1.08E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336489(1,2,4-trimethoxybenzene | CHEMBL1668605)
Affinity DataKi:  1.43E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataKi:  2.37E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50146462((2E)-3-(2-hydroxyphenyl)-2-propenoic acid | (2E)-3...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM36302(1,4-dimethoxybenzene)
Affinity DataKi:  3.35E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataKi:  3.53E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataKi:  3.67E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM36302(1,4-dimethoxybenzene)
Affinity DataKi:  4.02E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336489(1,2,4-trimethoxybenzene | CHEMBL1668605)
Affinity DataKi:  4.06E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50100861(3,4-Dihydroxybenzoate, VIII | 3,4-dihydroxybenzoic...)
Affinity DataKi:  4.09E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM36302(1,4-dimethoxybenzene)
Affinity DataKi:  4.15E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-DIHYDROXYBENZOATE | 3,5-Dihydroxy-benzoic acid...)
Affinity DataKi:  4.41E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50100861(3,4-Dihydroxybenzoate, VIII | 3,4-dihydroxybenzoic...)
Affinity DataKi:  4.45E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336491(3-Hydroxy-benzoic acid | 3-Hydroxybenzoate | 3-Hyd...)
Affinity DataKi:  4.53E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336489(1,2,4-trimethoxybenzene | CHEMBL1668605)
Affinity DataKi:  5.96E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336487(3,4-Dimethoxy-benzoic acid | 3,4-dimethoxybenzoic ...)
Affinity DataKi:  6.18E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336487(3,4-Dimethoxy-benzoic acid | 3,4-dimethoxybenzoic ...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336487(3,4-Dimethoxy-benzoic acid | 3,4-dimethoxybenzoic ...)
Affinity DataKi:  6.83E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336489(1,2,4-trimethoxybenzene | CHEMBL1668605)
Affinity DataKi:  7.80E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM36302(1,4-dimethoxybenzene)
Affinity DataKi:  8.21E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336492(2,6-dimethoxybenzoic acid | CHEMBL488609)
Affinity DataKi:  8.23E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336487(3,4-Dimethoxy-benzoic acid | 3,4-dimethoxybenzoic ...)
Affinity DataKi:  8.25E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336488(1,2-dimethoxybenzene | CHEMBL1668603)
Affinity DataKi:  8.36E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM10868(1,3,4-Thiadiazole-2-sulfonamide, 6 | 1,3,4-thiadia...)
Affinity DataKi:  8.60E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336488(1,2-dimethoxybenzene | CHEMBL1668603)
Affinity DataKi:  8.63E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336492(2,6-dimethoxybenzoic acid | CHEMBL488609)
Affinity DataKi:  9.07E+3nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50146462((2E)-3-(2-hydroxyphenyl)-2-propenoic acid | (2E)-3...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336492(2,6-dimethoxybenzoic acid | CHEMBL488609)
Affinity DataKi:  9.67E+3nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM26187(α-CA inhibitor, 11 | CHEMBL14060 | US9688816,...)
Affinity DataKi:  1.02E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50336488(1,2-dimethoxybenzene | CHEMBL1668603)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataKi:  1.33E+4nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataKi:  2.76E+4nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataKi:  8.40E+4nMAssay Description:Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM79403(3-aminopropyl-[4-(3-aminopropylamino)butyl]amine;h...)
Affinity DataKi:  2.31E+5nMAssay Description:Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50146462((2E)-3-(2-hydroxyphenyl)-2-propenoic acid | (2E)-3...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human carbonic anhydrase 12 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Calgary

Curated by ChEMBL
LigandPNGBDBM50146462((2E)-3-(2-hydroxyphenyl)-2-propenoic acid | (2E)-3...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins by CO2 hydration stopped-flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed