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Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50033039
TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338624((R)-3-amino-1-(3-(4-(methoxycarbonyl)phenyl)-6,7-d...)
Affinity DataIC50:  12.4nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338635((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(methox...)
Affinity DataIC50:  15.1nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338619((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(furan-...)
Affinity DataIC50:  15.8nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338615((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  17.8nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  19.4nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338637((R)-3-amino-1-(3-(difluoromethyl)-6,7-dihydro-[1,2...)
Affinity DataIC50:  22.5nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338617((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  22.8nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338618((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(furan-...)
Affinity DataIC50:  26.2nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338625((R)-3-amino-1-(3-(4-(dimethyamide)phenyl)-6,7-dihy...)
Affinity DataIC50:  26.6nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338621((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  28.6nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338634((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(amide)...)
Affinity DataIC50:  29.9nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338628((R)-3-amino-1-(3-(4-(cyano)phenyl)-6,7-dihydro-[1,...)
Affinity DataIC50:  30.0nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338622((R)-3-amino-1-(3-(4-(mesyl)phenyl)-6,7-dihydro-[1,...)
Affinity DataIC50:  33.2nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338620((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  33.3nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338623((R)-3-amino-1-(3-(4-(carboxyl)phenyl)-6,7-dihydro-...)
Affinity DataIC50:  33.8nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338626((R)-3-amino-1-(3-(4-(amide)phenyl)-6,7-dihydro-[1,...)
Affinity DataIC50:  36.4nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338632((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(4-phen...)
Affinity DataIC50:  37.5nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338631((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(4-fluo...)
Affinity DataIC50:  45.2nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338627((R)-3-amino-1-(3-(3-(methoxycarbonyl)phenyl)-6,7-d...)
Affinity DataIC50:  46.6nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338630((R)-3-amino-1-(3-(4-chlorophenyl)-6,7-dihydro-[1,2...)
Affinity DataIC50:  46.9nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338616((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  47.3nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338636((R)-3-amino-1-(3-(trifluoromethyl)-6,7-dihydro-[1,...)
Affinity DataIC50:  50.7nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338633((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(3-(dimeth...)
Affinity DataIC50:  52.3nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338629((R)-3-amino-1-(3-(4-(trifluoromethyl)phenyl)-6,7-d...)
Affinity DataIC50:  75.3nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338638((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  77.1nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDipeptidyl peptidase 4(Human)
Shandong University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50338639((R)-3-amino-4-(2,4,5-trifluorophenyl)-1-(6,7-dihyd...)
Affinity DataIC50:  89.5nMAssay Description:Inhibition of human DPP4 assessed as hydrolytic reaction of Ala-Pro-AMCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed