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Found 20 Enz. Inhib. hit(s) with all data for entry = 50033322
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343293(6-[5-(Cyclopropylmethyl)-4,5-dihydro-1'H,3H-spiro[...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343293(6-[5-(Cyclopropylmethyl)-4,5-dihydro-1'H,3H-spiro[...)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343291(CHEMBL1774095 | N-(2-Hydroxy-2-pyridin-3-ylethyl)-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343291(CHEMBL1774095 | N-(2-Hydroxy-2-pyridin-3-ylethyl)-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343290(6-(5-Ethyl-4,5-dihydro-1'H,3H-spiro[1,5-benzoxazep...)
Affinity DataIC50:  40nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50306110(CHEMBL607314 | N-(2-hydroxy-2-phenylethyl)-6-(4-ox...)
Affinity DataIC50:  50nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343288(CHEMBL1774092 | N-(2-hydroxy-2-phenylethyl)-6-(5-m...)
Affinity DataIC50:  50nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343290(6-(5-Ethyl-4,5-dihydro-1'H,3H-spiro[1,5-benzoxazep...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50306110(CHEMBL607314 | N-(2-hydroxy-2-phenylethyl)-6-(4-ox...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343288(CHEMBL1774092 | N-(2-hydroxy-2-phenylethyl)-6-(5-m...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343289(CHEMBL1774093 | N-(2-Hydroxy-2-pyridin-3-ylethyl)-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343294(6-[5-(2-Hydroxyethyl)-4,5-dihydro-1'H,3H-spiro[1,5...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343289(CHEMBL1774093 | N-(2-Hydroxy-2-pyridin-3-ylethyl)-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343287(6-(4,5-dihydro-3H-spiro[benzo[b][1,4]oxazepine-2,4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343286(CHEMBL1774090 | N-(2-hydroxy-2-phenylethyl)-6-(4-o...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343286(CHEMBL1774090 | N-(2-hydroxy-2-phenylethyl)-6-(4-o...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343285(CHEMBL1774089 | N-(2-hydroxy-2-(pyridin-3-yl)ethyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343287(6-(4,5-dihydro-3H-spiro[benzo[b][1,4]oxazepine-2,4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343294(6-[5-(2-Hydroxyethyl)-4,5-dihydro-1'H,3H-spiro[1,5...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343292(6-(5-Cyclopropyl-4,5-dihydro-1'H,3H-spiro[1,5-benz...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed