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Found 9 Enz. Inhib. hit(s) with all data for entry = 50033213
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341487(CHEMBL1765236 | Succinyl-alaninyl-alaninyl-proliny...)
Affinity DataIC50:  0.700nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated with alpha-chymotrypsin up to 8 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50:  1nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  1.5nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341488(CHEMBL1765235 | Phenylalaninyl-prolinyl-alaninyl-L...)
Affinity DataIC50:  7nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341488(CHEMBL1765235 | Phenylalaninyl-prolinyl-alaninyl-L...)
Affinity DataIC50:  8.30nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341489(CHEMBL1765234 | Cyclohexyl(glycinyl)-prolinyl-vali...)
Affinity DataIC50:  19nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341489(CHEMBL1765234 | Cyclohexyl(glycinyl)-prolinyl-vali...)
Affinity DataIC50:  20nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050513((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...)
Affinity DataIC50:  470nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University Sackler School Of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50:  1.60E+3nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed