Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50033118
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339823BDBM50339823(N-((2S)-3-(8',9'-dihydro-3'H-spiro[piperidine-3,7'...)
Affinity DataIC50: 9nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339824BDBM50339824(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6'-oxo-4',6...)
Affinity DataIC50: 10nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339825BDBM50339825(1'-((S)-3-(N-(2-ethoxyethyl)-2,6-dimethylphenylsul...)
Affinity DataIC50: 26nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339824BDBM50339824(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6'-oxo-4',6...)
Affinity DataIC50: 35nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339826BDBM50339826(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxysp...)
Affinity DataIC50: 40nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339823BDBM50339823(N-((2S)-3-(8',9'-dihydro-3'H-spiro[piperidine-3,7'...)
Affinity DataIC50: 44nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339827BDBM50339827(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxysp...)
Affinity DataIC50: 70nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339828BDBM50339828(N-((2S)-3-(6-cyanospiro[chroman-2,3'-piperidine]-1...)
Affinity DataIC50: 170nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339829BDBM50339829(N-(2-ethoxyethyl)-N-((2S)-3-(6-fluorospiro[chroman...)
Affinity DataIC50: 180nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339830BDBM50339830(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339831BDBM50339831(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339832BDBM50339832(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 500nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339834BDBM50339834(2-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339833BDBM50339833(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339835BDBM50339835(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339836BDBM50339836(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339825BDBM50339825(1'-((S)-3-(N-(2-ethoxyethyl)-2,6-dimethylphenylsul...)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339828BDBM50339828(N-((2S)-3-(6-cyanospiro[chroman-2,3'-piperidine]-1...)
Affinity DataIC50: 2.58E+3nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339826BDBM50339826(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxysp...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339838BDBM50339838(N-benzyl-N-(2-hydroxy-3-(6-hydroxy-4-oxospiro[chro...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339839BDBM50339839(N-cyclohexyl-N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxos...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339829BDBM50339829(N-(2-ethoxyethyl)-N-((2S)-3-(6-fluorospiro[chroman...)
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339840BDBM50339840(2-cyano-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-h...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339841BDBM50339841(N-(2-ethoxyethyl)-2-fluoro-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339827BDBM50339827(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxysp...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339831BDBM50339831(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339830BDBM50339830(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339844BDBM50339844(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339845BDBM50339845(4-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339843BDBM50339843(3-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339842BDBM50339842(N-((2R)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of AKT1 by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339842BDBM50339842(N-((2R)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339833BDBM50339833(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339835BDBM50339835(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339839BDBM50339839(N-cyclohexyl-N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxos...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339837BDBM50339837(N-((2S)-2-hydroxy-3-(6-hydroxy-4-oxospiro[chroman-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339841BDBM50339841(N-(2-ethoxyethyl)-2-fluoro-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339840BDBM50339840(2-cyano-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-h...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339836BDBM50339836(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339832BDBM50339832(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339843BDBM50339843(3-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339845BDBM50339845(4-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339834BDBM50339834(2-chloro-N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Array Biopharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339844BDBM50339844(N-(2-ethoxyethyl)-N-((2S)-2-hydroxy-3-(6-hydroxy-4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of AKT1 in human LNCaP cells assessed as PRAS40 phosphorylation at Thr246 after 1.5 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed