Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50033146
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340346BDBM50340346(2-(4-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50: 1nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340362BDBM50340362(2-(4-chloro-2-fluorophenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50: 1nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340341BDBM50340341(2-phenyl-1-{3-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50: 2nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340349BDBM50340349(2-(4-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50: 3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340360BDBM50340360(2-(2,4-dichlorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50: 3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340346BDBM50340346(2-(4-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50: 3nMAssay Description:Inhibition hERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340363BDBM50340363(2-(3,4-difluorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50: 4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340364BDBM50340364(2-(2-chloro-4-fluorophenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50: 4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340345BDBM50340345(2-(3-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50: 5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340367BDBM50340367(2-(4-chlorophenyl)-1-{3-[4-(3-isobutyrylaminopheny...)
Affinity DataIC50: 5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340354BDBM50340354(2-(4-bromophenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50: 5nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340351BDBM50340351(2-(3-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50: 7nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340357BDBM50340357(2-(4-biphenyl)-1-{3-[4-(3-acetylaminophenyl)piperi...)
Affinity DataIC50: 8nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340352BDBM50340352(2-(4-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50: 9nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340344BDBM50340344(2-(2-chlorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50: 10nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340359BDBM50340359(2-(4-cyanophenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50: 16nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340368BDBM50340368(2-(4-chlorophenyl)-1-{3-[4-(3-benzoylaminophenyl)p...)
Affinity DataIC50: 19nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340361BDBM50340361(2-(3,4-dichlorophenyl)-1-{3-[4-(3-acetylaminopheny...)
Affinity DataIC50: 24nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340342BDBM50340342(2-phenyl-1-{4-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50: 29nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340348BDBM50340348(2-(3-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50: 30nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340355BDBM50340355(2-(4-Ethylphenyl)-1-{3-[4-(3-acetylaminophenyl)pip...)
Affinity DataIC50: 32nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340358BDBM50340358(2-(4-phenoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50: 42nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340347BDBM50340347(2-(2-trifluoromethylphenyl)-1-{3-[4-(3-acetylamino...)
Affinity DataIC50: 50nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340353BDBM50340353(2-(4-Fluorophenyl)-1-{3-[4-(3-acetylaminophenyl)pi...)
Affinity DataIC50: 56nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340356BDBM50340356(2-(4-isopropylphenyl)-1-{3-[4-(3-acetylaminophenyl...)
Affinity DataIC50: 60nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340343BDBM50340343(2-phenyl-1-{5-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50: 74nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340370BDBM50340370(2-(4-chlorophenyl)-1-{3-[4-(3-(4-methylbenzoylamin...)
Affinity DataIC50: 213nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340369BDBM50340369(2-(4-chlorophenyl)-1-{3-[4-(3-(3-chlorobenzoylamin...)
Affinity DataIC50: 300nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340350BDBM50340350(2-(2-methoxyphenyl)-1-{3-[4-(3-acetylaminophenyl)p...)
Affinity DataIC50: 747nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340366BDBM50340366(2-(4-chlorophenyl)-1-{5-[4-(4-acetylaminophenyl)pi...)
Affinity DataIC50: 5.38E+3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340365BDBM50340365(2-(4-chlorophenyl)-1-{5-[4-(2-acetylaminophenyl)pi...)
Affinity DataIC50: 6.00E+3nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340340BDBM50340340(2-phenyl-1-{2-[4-(3-acetylaminophenyl)piperidin-1-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of Eu-labeled MCH from human MCH-R1 expressed in CHO by time-resolved fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed