Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50001127
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013025(CHEMBL305903 | 2,6-Dimethyl-4-(5-methyl-3-phenyl-i...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013025(CHEMBL305903 | 2,6-Dimethyl-4-(5-methyl-3-phenyl-i...)
Affinity DataKi:  22nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013022(CHEMBL74944 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013022(CHEMBL74944 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013022(CHEMBL74944 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013022(CHEMBL74944 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  33nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013021(CHEMBL72620 | 4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2...)
Affinity DataKi:  52nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013021(CHEMBL72620 | 4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2...)
Affinity DataKi:  63nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013026(CHEMBL72717 | 2,6-Dimethyl-4-(5-pentyl-3-phenyl-is...)
Affinity DataKi:  78nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013026(CHEMBL72717 | 2,6-Dimethyl-4-(5-pentyl-3-phenyl-is...)
Affinity DataKi:  79nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013024(CHEMBL73647 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  122nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013024(CHEMBL73647 | 4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-d...)
Affinity DataKi:  173nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50013023(CHEMBL75770 | 4-(5-Isopropyl-3-phenyl-isoxazol-4-y...)
Affinity DataKi:  254nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50013023(CHEMBL75770 | 4-(5-Isopropyl-3-phenyl-isoxazol-4-y...)
Affinity DataKi:  417nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed