Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50033151
TargetDipeptidyl peptidase 4(Human)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340427(1-((3S,8S,9S,10R,13S,14S,17R)-16-(benzylamino)-3-h...)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340428(3-(3,4-dimethoxyphenyl)-1-((3S,8R,9S,10R,13S,14S)-...)
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340430((2S,4aR,4bS,6aS,9R,11aS,11bS)-2-Hydroxy-9-(4-isopr...)
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340429((2S,4aR,4bS,6aS,9R,11aS,11bS)-2-Hydroxy-9-(4-metho...)
Affinity DataIC50: 3.27E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340426(16-Dehydropregnenolone acetate | CHEMBL1761683)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed