Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50041908
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12746BDBM12746(6-[4-(2-methanesulfonylphenyl)phenyl]-1-(4-methoxy...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 12743BDBM12743(6-[4-(2-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phe...)
Affinity DataKi:  0.501nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13286BDBM13286(4-hydroxy-3-{[(3S)-3-[(7-methoxynaphthalene-2-)sul...)
Affinity DataKi:  3.16nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081002BDBM50081002(4-Amino-3-[3-((S)-7-methoxy-naphthalene-2-sulfonyl...)
Affinity DataKi:  6.31nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19018BDBM19018(6-[4-(dimethylamino)phenyl]-1-(4-methoxyphenyl)-3-...)
Affinity DataKi:  6.31nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13288BDBM13288(methyl 2-(4-carbamimidoyl-2-{[(3S)-3-[(7-methoxyna...)
Affinity DataKi:  7.94nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13668BDBM13668(4-chloro-3-[2-(4-chlorophenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  12.6nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13615BDBM13615(4-chloro-3-[2-(5-chloropyridin-2-yl)ethoxy]-N-{[1-...)
Affinity DataKi:  19.9nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13667BDBM13667(4-chloro-3-[2-(2,4-dichlorophenyl)ethoxy]-N-{[1-(p...)
Affinity DataKi:  39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13619BDBM13619(3-[2-(4-bromophenyl)ethoxy]-4-chloro-N-{[1-(pyridi...)
Affinity DataKi:  39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13618BDBM13618(3-[2-(5-chloropyridin-2-yl)ethoxy]-4-fluoro-N-{[1-...)
Affinity DataKi:  39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13617BDBM13617(3-[2-(4-chlorophenyl)ethoxy]-4-fluoro-N-{[1-(pyrid...)
Affinity DataKi:  39.8nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13616BDBM13616(3-[2-(2,4-dichlorophenyl)ethoxy]-4-fluoro-N-{[1-(p...)
Affinity DataKi:  50.1nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50081006BDBM50081006(3-[3-((S)-7-Methoxy-naphthalene-2-sulfonylamino)-2...)
Affinity DataKi:  50.1nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13629BDBM13629(3-[2-(4-bromophenyl)ethoxy]-4-fluoro-N-{[1-(pyridi...)
Affinity DataKi:  79.4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13620BDBM13620(4-chloro-3-[2-(4-fluorophenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  100nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13621BDBM13621(4-chloro-3-[2-(4-methylphenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  126nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13631BDBM13631(4-fluoro-3-[2-(4-methylphenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13630BDBM13630(4-fluoro-3-[2-(4-fluorophenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19015BDBM19015(N-{4-[1-(4-methoxyphenyl)-7-oxo-3-(trifluoromethyl...)
Affinity DataKi:  200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13632BDBM13632(4-fluoro-3-[2-(4-methoxyphenyl)ethoxy]-N-{[1-(pyri...)
Affinity DataKi:  316nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13622BDBM13622(4-chloro-3-[2-(4-methoxyphenyl)ethoxy]-N-{[1-(pyri...)
Affinity DataKi:  316nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13626BDBM13626(3-[2-(4-aminophenyl)ethoxy]-4-chloro-N-{[1-(pyridi...)
Affinity DataKi:  398nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13634BDBM13634(3-[2-(3-chlorophenyl)ethoxy]-4-fluoro-N-{[1-(pyrid...)
Affinity DataKi:  631nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13287BDBM13287(2-hydroxy-5-{[(3S)-3-[(7-methoxynaphthalene-2-)sul...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13285BDBM13285(3-Amino-5-[3-(S)-(7-methoxynaphthalen-2-ylsulfonyl...)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418332BDBM50418332(CHEMBL1766822)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13636BDBM13636(3-[2-(4-aminophenyl)ethoxy]-4-fluoro-N-{[1-(pyridi...)
Affinity DataKi:  1.58E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13623BDBM13623(4-chloro-3-[2-(4-cyanophenyl)ethoxy]-N-{[1-(pyridi...)
Affinity DataKi:  1.58E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 19014BDBM19014(6-(4-aminophenyl)-1-(4-methoxyphenyl)-3-(trifluoro...)
Affinity DataKi:  1.58E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13624BDBM13624(4-chloro-3-[2-(3-chlorophenyl)ethoxy]-N-{[1-(pyrid...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13625BDBM13625(4-chloro-3-[2-(3-methoxyphenyl)ethoxy]-N-{[1-(pyri...)
Affinity DataKi:  2.51E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13635BDBM13635(4-fluoro-3-[2-(3-methoxyphenyl)ethoxy]-N-{[1-(pyri...)
Affinity DataKi:  3.16E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13633BDBM13633(3-[2-(4-cyanophenyl)ethoxy]-4-fluoro-N-{[1-(pyridi...)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13627BDBM13627(tert-butyl N-(4-{2-[2-chloro-5-({[1-(pyridin-4-yl)...)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13638BDBM13638(3-[2-(4-acetamidophenyl)ethoxy]-4-fluoro-N-{[1-(py...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13637BDBM13637(tert-butyl N-(4-{2-[2-fluoro-5-({[1-(pyridin-4-yl)...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rheinische Friedrich-Wilhelms-Universita£T

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13628BDBM13628(4-chloro-3-[2-(4-acetamidophenyl)ethoxy]-N-{[1-(py...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed