Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50004524
TargetReverse transcriptase(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50:  223nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50:  223nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50369390(CHEMBL54224)
Affinity DataIC50:  244nMAssay Description:Inhibition of HIV-1 reverse transcriptase K101E mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50175609(5-{3-[4-Amino-9-(tert-butyl-dimethyl-silanyloxy)-6...)
Affinity DataIC50:  560nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50169035(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50483735(CHEMBL1766951)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of wild type HIV-1 reverse transcriptase-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: >1.65E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase K101E mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50192289(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: >1.65E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Rutgers University

Curated by ChEMBL
LigandPNGBDBM50169035(1-[(5R,6R,8R,9R)-4-amino-9-(tert-butyl-dimethyl-si...)
Affinity DataIC50: >1.69E+5nMAssay Description:Inhibition of HIV-1 reverse transcriptase E138K mutant-mediated polymerization reaction after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed