Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50033340
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002087BDBM50002087(4-(1-Methyl-piperidin-4-ylidene)-4,9-dihydro-1-thi...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295709BDBM50295709(2-(10-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrah...)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343578BDBM50343578(5-(3-(4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro...)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343589BDBM50343589(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 54nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343583BDBM50343583((Z)-11-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetra...)
Affinity DataIC50: 63nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343572BDBM50343572(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro...)
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343588BDBM50343588(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 75nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22874BDBM22874(CHEMBL914 | Allegra | 2-(4-{1-hydroxy-4-[4-(hydrox...)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343587BDBM50343587((Z)-2-(11-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-te...)
Affinity DataIC50: 84nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343585BDBM50343585((Z)-2-(11-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-te...)
Affinity DataIC50: 92nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343576BDBM50343576(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 128nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343575BDBM50343575(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 128nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343581BDBM50343581([(5Z)-5-{3-[4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetr...)
Affinity DataIC50: 135nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343579BDBM50343579(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro...)
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343574BDBM50343574(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343580BDBM50343580((5Z)-5-{3-[4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetra...)
Affinity DataIC50: 153nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343582BDBM50343582([(5Z)-5-{3-[4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetr...)
Affinity DataIC50: 195nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343577BDBM50343577(2-(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahy...)
Affinity DataIC50: 255nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343584BDBM50343584((Z)-11-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetra...)
Affinity DataIC50: 325nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343573BDBM50343573(5-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro...)
Affinity DataIC50: 530nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343586BDBM50343586((E)-2-(11-(3-(4-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-te...)
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO-K1 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed