Affinity DataIC50: 158nMAssay Description:Antagonist activity at FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated degranulation after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Antagonist activity at human FPR1 in expressed in HEK293 cells assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation after 5 m...More data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at FPR1More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+3nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+4nMAssay Description:Antagonist activity at mouse FPR1 expressed in HEK293 cells assessed as inhibition of fMLFF-stimulated intracellular calcium mobilisation by FLIPR as...More data for this Ligand-Target Pair