Compile Data Set for Download or QSAR
maximum 50k data
Found 87 Enz. Inhib. hit(s) with all data for entry = 50033443
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50341879(CHEMBL1767408 | Diquafosol)
Affinity DataEC50:  1.31E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271251(CHEMBL483502 | {[({[({[(2R,3S,4R,5R)-5-(2,4-dioxo-...)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271291(CHEMBL484105 | Uridine-5'-(2-cyanoethyl)-tetraphos...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270541(CHEMBL474886 | Uridine-5'-phenyl-tetraphosphate)
Affinity DataEC50:  1.89E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345483(CHEMBL1784891 | N4-t-Butyloxycytidine-5'-triphosph...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345484(CHEMBL1784892 | N4-Benzyloxycytidine-5'-triphospha...)
Affinity DataEC50:  620nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345485(CHEMBL1784893 | N4-Phenylethoxycytidine-5'-triphos...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345486(CHEMBL1784894 | N4-Phenylpropoxycytidine-5'-tripho...)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345480(((2R,3S,4R,5R)-4-azido-5-(2,4-dioxo-3,4-dihydropyr...)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270541(CHEMBL474886 | Uridine-5'-phenyl-tetraphosphate)
Affinity DataEC50:  2.76E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345494(CHEMBL1784889 | P1-(Uridine-5'-)P4-(2'-deoxy-2'-ac...)
Affinity DataEC50:  1.89E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345482(CHEMBL1784890 | N4-Ethoxycytidine-5'-triphosphate)
Affinity DataEC50:  817nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271187(CHEMBL519835 | [dichloro({[({[(2R,3S,4R,5R)-3,4-di...)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50319143(CHEMBL1083764 | CHEMBL1198849 | N4-Methoxycytidine...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345491(CHEMBL1784885 | Uridine-5'-allose-1'-tetraphosphat...)
Affinity DataEC50:  770nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345492(CHEMBL1784886 | Uridine-5'-mannose-1'-tetraphospha...)
Affinity DataEC50:  3.72E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345493(CHEMBL1784887 | Uridine-5'-xylose-1'-tetraphosphat...)
Affinity DataEC50:  2.77E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271187(CHEMBL519835 | [dichloro({[({[(2R,3S,4R,5R)-3,4-di...)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270546(CHEMBL444212 | Uridine-5'-galactose-1'-tetraphosph...)
Affinity DataEC50:  940nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(CHEMBL499138 | Uridine-5'-glucose-1'-tetraphosphat...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50205406(((2R,3S,4R,5R)-4-amino-3-hydroxy-5-(4-oxo-2-thioxo...)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345495(CHEMBL1784902 | P1-(Uridine-5'-)P4-(glucuronic aci...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345496(CHEMBL1784904 | P1-(Uridine-5'-)P4-(3'-deoxy-3'-fl...)
Affinity DataEC50:  710nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270551(CHEMBL502712 | P1,P4-di(uridine 5'-)beta,gamma-dif...)
Affinity DataEC50:  2.27E+3nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50271289(CHEMBL519991 | Uridine-5'-methyl-tetraphosphate)
Affinity DataEC50:  4.00E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345489(CHEMBL1784899 | Uridine-5'-(4-nitrophenyl)-tetraph...)
Affinity DataEC50:  4.85E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345490(CHEMBL1784900 | Uridine-5'-(3-nitrophenyl)-tetraph...)
Affinity DataEC50:  3.33E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(CHEMBL499138 | Uridine-5'-glucose-1'-tetraphosphat...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345487(CHEMBL1784895 | Uridine-5'-(4-chlorophenyl)-tetrap...)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345498(CHEMBL1784292 | P1-(N4-Methoxycytidine-5'-)P4-(3'-...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345488(CHEMBL1784896 | Uridine-5'-(3-chlorophenyl)-tetrap...)
Affinity DataEC50:  840nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345497(CHEMBL1784291 | P1-(N4-Benzyloxycytidine-5'-)P4-(3...)
Affinity DataEC50:  2.64E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human P2Y2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50341896(CHEMBL1765114 | dichloro(((((2R,3S,4R,5R)-5-(2,4-d...)
Affinity DataEC50:  9.60E+3nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345499(CHEMBL1784293 | P1-(Uridine-5'-)P4-(4'-deoxy-4'-fl...)
Affinity DataEC50:  620nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50341879(CHEMBL1767408 | Diquafosol)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50341879(CHEMBL1767408 | Diquafosol)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345480(((2R,3S,4R,5R)-4-azido-5-(2,4-dioxo-3,4-dihydropyr...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(5'-UTP | CHEMBL336296 | H4utp | UTP | uridine 5'-(...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50341879(CHEMBL1767408 | Diquafosol)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50270545(CHEMBL499138 | Uridine-5'-glucose-1'-tetraphosphat...)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50319143(CHEMBL1083764 | CHEMBL1198849 | N4-Methoxycytidine...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345482(CHEMBL1784890 | N4-Ethoxycytidine-5'-triphosphate)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345483(CHEMBL1784891 | N4-t-Butyloxycytidine-5'-triphosph...)
Affinity DataEC50:  2.11E+3nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345484(CHEMBL1784892 | N4-Benzyloxycytidine-5'-triphospha...)
Affinity DataEC50:  97nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50345485(CHEMBL1784893 | N4-Phenylethoxycytidine-5'-triphos...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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