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Found 24 Enz. Inhib. hit(s) with all data for entry = 50033574
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347558(CHEMBL1802233)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347560(CHEMBL1802235)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347557(CHEMBL1802232)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347562(CHEMBL1802237)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347557(CHEMBL1802232)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347561(CHEMBL1802236)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347556(CHEMBL1802231)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347560(CHEMBL1802235)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347561(CHEMBL1802236)
Affinity DataKi:  400nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347562(CHEMBL1802237)
Affinity DataKi:  415nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347559(CHEMBL1802234)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]raclopride from rat D2 dopamine receptor expressed in CHOK1 cells after 90 mins by liquid scintillation counter scintillation cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347558(CHEMBL1802233)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347559(CHEMBL1802234)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347556(CHEMBL1802231)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347556(CHEMBL1802231)
Affinity DataEC50:  211nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347562(CHEMBL1802237)
Affinity DataEC50:  383nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347561(CHEMBL1802236)
Affinity DataEC50:  148nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347560(CHEMBL1802235)
Affinity DataEC50:  24nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347559(CHEMBL1802234)
Affinity DataEC50:  820nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347558(CHEMBL1802233)
Affinity DataEC50:  16nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50347557(CHEMBL1802232)
Affinity DataEC50:  198nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Tartu

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed