Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50033699
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM23738(2-(1-benzyl-5-methoxy-2-methyl-1H-indol-3-yl)aceta...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349888(CHEMBL1814415)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349880(CHEMBL1814402)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349890(CHEMBL1814417)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349883(CHEMBL1814409)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349882(CHEMBL1814404)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349881(CHEMBL1814403)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349884(CHEMBL1814410)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349879(CHEMBL1814401)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349886(CHEMBL1814412)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349891(CHEMBL1814418)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349885(CHEMBL1814411)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349892(CHEMBL1814419)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349887(CHEMBL1814414)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349889(CHEMBL1814416)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Peking University

Curated by ChEMBL
LigandPNGBDBM50349893(CHEMBL1814420)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of human non-pancreatic sPLA2 using 1,2-dimyristoyl-sn-glycero-3-phosphocholine substrate after 5 mins by continuous fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed