Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50033701
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11639BDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140317BDBM50140317((R)-2-[4-((1R,2S)-2-Hydroxy-cyclopentylmethyl)-phe...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349898BDBM50349898(CHEMBL1814707)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140317BDBM50140317((R)-2-[4-((1R,2S)-2-Hydroxy-cyclopentylmethyl)-phe...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349898BDBM50349898(CHEMBL1814707)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349902BDBM50349902(CHEMBL1814711)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 11639BDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330853BDBM50330853(Sodium; 2-[4-(2-oxo-cyclopentylmethyl)-phenyl]-pro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349918BDBM50349918(CHEMBL1814726)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349902BDBM50349902(CHEMBL1814711)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330851BDBM50330851(fluoro loxoprofen | CHEMBL1275921)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349920BDBM50349920(CHEMBL1814728)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349919BDBM50349919(CHEMBL1814727)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349901BDBM50349901(CHEMBL1814710)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330853BDBM50330853(Sodium; 2-[4-(2-oxo-cyclopentylmethyl)-phenyl]-pro...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330851BDBM50330851(fluoro loxoprofen | CHEMBL1275921)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330850BDBM50330850(bromoloxoprofen | CHEMBL1275940)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349907BDBM50349907(CHEMBL1814716)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349915BDBM50349915(CHEMBL1814724)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349920BDBM50349920(CHEMBL1814728)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349900BDBM50349900(CHEMBL1814709)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349901BDBM50349901(CHEMBL1814710)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349903BDBM50349903(CHEMBL1814712)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349904BDBM50349904(CHEMBL1814713)
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50330850BDBM50330850(bromoloxoprofen | CHEMBL1275940)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349911BDBM50349911(CHEMBL1814720)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349908BDBM50349908(CHEMBL1814717)
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349913BDBM50349913(CHEMBL1814722)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349917BDBM50349917(CHEMBL1814725)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349900BDBM50349900(CHEMBL1814709)
Affinity DataIC50: 9.30E+4nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349914BDBM50349914(CHEMBL1814723)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349915BDBM50349915(CHEMBL1814724)
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349907BDBM50349907(CHEMBL1814716)
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349899BDBM50349899(CHEMBL1814708)
Affinity DataIC50: 2.70E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349903BDBM50349903(CHEMBL1814712)
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349911BDBM50349911(CHEMBL1814720)
Affinity DataIC50: 3.10E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349918BDBM50349918(CHEMBL1814726)
Affinity DataIC50: 3.26E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349904BDBM50349904(CHEMBL1814713)
Affinity DataIC50: 4.20E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349913BDBM50349913(CHEMBL1814722)
Affinity DataIC50: 4.30E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349908BDBM50349908(CHEMBL1814717)
Affinity DataIC50: 4.60E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349912BDBM50349912(CHEMBL1814721)
Affinity DataIC50: 4.70E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349916BDBM50349916(CHEMBL1814706)
Affinity DataIC50: 5.15E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349912BDBM50349912(CHEMBL1814721)
Affinity DataIC50: 5.40E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349899BDBM50349899(CHEMBL1814708)
Affinity DataIC50: 5.40E+5nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349914BDBM50349914(CHEMBL1814723)
Affinity DataIC50: 5.75E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349919BDBM50349919(CHEMBL1814727)
Affinity DataIC50: 6.50E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349906BDBM50349906(CHEMBL1814715)
Affinity DataIC50: 7.58E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349905BDBM50349905(CHEMBL1814714)
Affinity DataIC50: 8.00E+5nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349909BDBM50349909(CHEMBL1814718)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human whole blood COX-2 assessed as production of PGE2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Kumamoto University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349917BDBM50349917(CHEMBL1814725)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human whole blood COX-1 assessed as production of TXB2 after 24 hrs by EIAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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