Compile Data Set for Download or QSAR
Report error Found 108 Enz. Inhib. hit(s) with all data for entry = 50033590
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347798BDBM50347798(CHEMBL1802410)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347802BDBM50347802(CHEMBL1802406)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347793BDBM50347793(CHEMBL1802966)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347793BDBM50347793(CHEMBL1802966)
Affinity DataIC50: 34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347792BDBM50347792(CHEMBL1802967)
Affinity DataIC50: 39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347815BDBM50347815(CHEMBL1802405)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347792BDBM50347792(CHEMBL1802967)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347796BDBM50347796(CHEMBL1802963)
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347802BDBM50347802(CHEMBL1802406)
Affinity DataIC50: 66nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347803BDBM50347803(CHEMBL1802404)
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347796BDBM50347796(CHEMBL1802963)
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347806BDBM50347806(CHEMBL1802401)
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347799BDBM50347799(CHEMBL1802409)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347806BDBM50347806(CHEMBL1802401)
Affinity DataIC50: 85nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347814BDBM50347814(CHEMBL1802391)
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347803BDBM50347803(CHEMBL1802404)
Affinity DataIC50: 95nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347798BDBM50347798(CHEMBL1802410)
Affinity DataIC50: 110nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347804BDBM50347804(CHEMBL1802403)
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10841BDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10841BDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347794BDBM50347794(CHEMBL1802965)
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347814BDBM50347814(CHEMBL1802391)
Affinity DataIC50: 190nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347799BDBM50347799(CHEMBL1802409)
Affinity DataIC50: 220nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10840BDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347804BDBM50347804(CHEMBL1802403)
Affinity DataIC50: 250nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347788BDBM50347788(CHEMBL1802971)
Affinity DataIC50: 290nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10840BDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347794BDBM50347794(CHEMBL1802965)
Affinity DataIC50: 330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347788BDBM50347788(CHEMBL1802971)
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347807BDBM50347807(CHEMBL1802400)
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347815BDBM50347815(CHEMBL1802405)
Affinity DataIC50: 460nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10844BDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347785BDBM50347785(CHEMBL1802390)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347800BDBM50347800(CHEMBL1802408)
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347798BDBM50347798(CHEMBL1802410)
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347793BDBM50347793(CHEMBL1802966)
Affinity DataIC50: 680nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10844BDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50: 700nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347786BDBM50347786(CHEMBL1802389)
Affinity DataIC50: 750nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347810BDBM50347810(CHEMBL1802396)
Affinity DataIC50: 810nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347808BDBM50347808(CHEMBL1802399)
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347797BDBM50347797(CHEMBL1802962)
Affinity DataIC50: 850nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347808BDBM50347808(CHEMBL1802399)
Affinity DataIC50: 870nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347801BDBM50347801(CHEMBL1802407)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347807BDBM50347807(CHEMBL1802400)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10841BDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10840BDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347811BDBM50347811(CHEMBL1802395)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347817BDBM50347817(CHEMBL1802392)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347810BDBM50347810(CHEMBL1802396)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Clermont Universite£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347797BDBM50347797(CHEMBL1802962)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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