Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50035892
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013761(CHEMBL3038194 | (R)-1-(3-cyclopropylmethyl-11,15-d...)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013388(CHEMBL350384 | BREMAZOCINE(-) | 6-Ethyl-3-(1-hydro...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50406411(CHEMBL2021332)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013764(CHEMBL3038199 | 5-(3-cyclopropylmethyl-11-hydroxy-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-ox...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataIC50: 5nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013763(CHEMBL3038197 | (S)-19-(1-isothiocyanatoethyl)-15-...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013768(CHEMBL3038193 | 3-O-(tert-Butyldimethylsilyl)-6,14...)
Affinity DataIC50: 34nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50406413(CHEMBL2021335)
Affinity DataIC50: 63nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013769(CHEMBL3038198 | (S)-1-(3-cyclopropylmethyl-11,15-d...)
Affinity DataIC50: 171nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013766(CHEMBL3038195 | (S)-1-(11,15-dimethoxy-3-methyl-13...)
Affinity DataIC50: 323nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50406412(CHEMBL2021333)
Affinity DataIC50: 434nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Bovine)
University of Washington

Curated by ChEMBL
LigandPNGBDBM50013760(CHEMBL3038196 | (R)-1-(11,15-dimethoxy-3-methyl-13...)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed