Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 50040370
TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393167(CHEMBL2153721)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50004587(8-Adamantan-1-yl-1,3-dipropyl-3,7-dihydro-purine-2...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  5.15nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50084860(3-(3-Hydroxy-propyl)-8-[2-(3-methoxy-phenyl)-vinyl...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  90.8nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393188(CHEMBL2153620)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393167(CHEMBL2153721)
Affinity DataKi:  269nMAssay Description:Displacement of [125I]ZM241385 from adenosine A2A receptor in rat brain striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393192(CHEMBL2153629)
Affinity DataKi:  306nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393192(CHEMBL2153629)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393172(CHEMBL2153627)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393181(CHEMBL2153614)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393189(CHEMBL2153612)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393188(CHEMBL2153620)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393177(CHEMBL2153618)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393192(CHEMBL2153629)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393191(CHEMBL2153624)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393187(CHEMBL2153607)
Affinity DataKi:  830nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393193(CHEMBL2153626)
Affinity DataKi:  847nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393180(CHEMBL2153615)
Affinity DataKi:  887nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50084860(3-(3-Hydroxy-propyl)-8-[2-(3-methoxy-phenyl)-vinyl...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393181(CHEMBL2153614)
Affinity DataKi:  933nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393172(CHEMBL2153627)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393173(CHEMBL2153625)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393176(CHEMBL2153619)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50004587(8-Adamantan-1-yl-1,3-dipropyl-3,7-dihydro-purine-2...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CGS21680 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393182(CHEMBL2153613)
Affinity DataKi:  1.16E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393197(CHEMBL2153604)
Affinity DataKi:  1.17E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393199(CHEMBL2153628)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393178(CHEMBL2153617)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A3(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393183(CHEMBL2153611)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393179(CHEMBL2153616)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393184(CHEMBL2151065)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393189(CHEMBL2153612)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393167(CHEMBL2153721)
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [3H]MRS-1754 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393191(CHEMBL2153624)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393169(CHEMBL2153632)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393197(CHEMBL2153604)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A3(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393190(CHEMBL2153603)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393186(CHEMBL2153608)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393193(CHEMBL2153626)
Affinity DataKi:  1.93E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393198(CHEMBL2153719)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393170(CHEMBL2153630)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393174(CHEMBL2153623)
Affinity DataKi:  2.04E+3nMAssay Description:Displacement of [3H]MSX-2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  2.07E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393185(CHEMBL2153610)
Affinity DataKi:  2.13E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393172(CHEMBL2153627)
Affinity DataKi:  2.39E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393190(CHEMBL2153603)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393170(CHEMBL2153630)
Affinity DataKi:  2.45E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Rat)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50393177(CHEMBL2153618)
Affinity DataKi:  2.49E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Displayed 1 to 50 (of 142 total ) | Next | Last >>
Jump to: