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Found 25 Enz. Inhib. hit(s) with all data for entry = 50033717
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM78304(2-(2-hydroxy-5-prop-2-enylphenyl)-4-prop-2-enylphe...)
Affinity DataEC50:  3.68E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM81563(Magreth-16a)
Affinity DataEC50:  1.43E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM81559(Magreth-11b)
Affinity DataEC50:  1.69E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM81558(Magreth-11a)
Affinity DataEC50:  8.40E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419019(CHEMBL1814294)
Affinity DataEC50:  2.00E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50350149(CHEMBL1814312)
Affinity DataEC50:  3.80E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419020(CHEMBL1814309)
Affinity DataEC50:  1.85E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419021(CHEMBL1814308)
Affinity DataEC50:  9.30E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419022(CHEMBL1814306)
Affinity DataEC50:  1.24E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419023(CHEMBL1814305)
Affinity DataEC50:  2.50E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419024(CHEMBL1814300)
Affinity DataEC50:  2.20E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM81565(Magreth-17a)
Affinity DataEC50:  1.48E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM81564(Magreth-16b)
Affinity DataEC50:  5.99E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50295927(2,4'-Dimethoxy-5,3'-di-(2-propenyl)-biphenyl | 5,3...)
Affinity DataEC50:  4.21E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419025(CHEMBL1814295)
Affinity DataEC50:  5.43E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419026(CHEMBL231391)
Affinity DataEC50:  2.37E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419027(CHEMBL182529)
Affinity DataEC50:  3.52E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419028(CHEMBL1814293)
Affinity DataEC50:  1.05E+5nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419029(CHEMBL1814291)
Affinity DataEC50:  3.42E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50295924(4'-Methoxy-3'-(Z)-propenyl)-5-(2-propenyl)-bipheny...)
Affinity DataEC50:  1.97E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50295920(4'-Methoxy-5,3'-dipropyl-biphenyl-2ol | CHEMBL5552...)
Affinity DataEC50:  1.27E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50419030(CHEMBL1814310)
Affinity DataEC50:  7.70E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50350150(CHEMBL1814307)
Affinity DataEC50:  9.20E+3nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50295926(4'-O-methylhonokiol, MH | 4-methoxyhonokiol | ...)
Affinity DataEC50:  2.72E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50157304(3',5-di-2-propenyl-1,1'-biphenyl-2,4'-diol | 3',5-...)
Affinity DataEC50:  3.93E+4nMAssay Description:Modulation of GABA Aalpha1beta2 receptor expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chloride current at holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed