Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50004559
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 1434BDBM1434(BI-RG-587 | 2-cyclopropyl-7-methyl-2,4,9,15-tetraa...)
Affinity DataIC50: 670nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2184BDBM2184(SM30 | US8501787, 166)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2173BDBM2173(CW23836 | US8501787, 116)
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2172BDBM2172(DG 402-49748 | US8501787, 104)
Affinity DataIC50: 3.74E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2115BDBM2115(MLB133-641A | US8501787, 8)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2116BDBM2116(DG 402-49706 | US8501787, 42)
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2177BDBM2177(SM27 | US8501787, 163)
Affinity DataIC50: 5.39E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 99893BDBM99893(US8501767, 96)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2182BDBM2182(SM29 | US8501787, 165)
Affinity DataIC50: 7.18E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2162BDBM2162(DG 402-49754 | US8501787, 97)
Affinity DataIC50: 7.52E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 99895BDBM99895(US8501767, 81)
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 99896BDBM99896(US8501767, 99)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 99894BDBM99894(US8501767, 82)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484067BDBM50484067(CHEMBL1807349)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed