Compile Data Set for Download or QSAR
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Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50001228
TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013943(CHEMBL327270 | Furan-2-carboxylic acid (2-chloro-p...)
Affinity DataKi:  0.130nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013945(CHEMBL431047 | Furan-2-carboxylic acid [3-methyl-1...)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013934(CHEMBL319060 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  0.190nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.220nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013939(CHEMBL95247 | Furan-2-carboxylic acid (3-methyl-1-...)
Affinity DataKi:  0.300nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013938(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013938(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  0.330nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013949(CHEMBL95248 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  0.780nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013948(CHEMBL95909 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013947(CHEMBL95786 | Furan-2-carboxylic acid (2-methoxy-p...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013935(CHEMBL95390 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-m...)
Affinity DataKi:  2nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013940(CHEMBL319343 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-...)
Affinity DataKi:  2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013942(CHEMBL318895 | N-(2-Chloro-phenyl)-2-methoxy-N-(3-...)
Affinity DataKi:  2.80nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013936(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013936(2-Methoxy-N-(3-methyl-1-phenethyl-piperidin-4-yl)-...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013944(2-Methoxy-N-(2-methoxy-phenyl)-N-(3-methyl-1-phene...)
Affinity DataKi:  7.60nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013941(CHEMBL99596 | N-(2-Fluoro-phenyl)-2-methoxy-N-(3-m...)
Affinity DataKi:  8.10nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM83450(ALFENTANIL | Alfentanil hydrochloride | MLS0023206...)
Affinity DataKi:  8.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013937(2-Methoxy-N-(2-methoxy-phenyl)-N-[3-methyl-1-(2-th...)
Affinity DataKi:  11nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013946(CHEMBL316670 | Furan-2-carboxylic acid (2-methoxy-...)
Affinity DataKi: >100nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Rat)
Anaquest Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50013935(CHEMBL95390 | N-(2-Fluoro-phenyl)-2-methoxy-N-[3-m...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed