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Found 17 Enz. Inhib. hit(s) with all data for entry = 50033768
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50350947(CHEMBL1818218)
Affinity DataIC50:  580nMAssay Description:Inhibition of human ERG expressed in human HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350947(CHEMBL1818218)
Affinity DataEC50:  97nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350948(CHEMBL1818217)
Affinity DataEC50:  109nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350947(CHEMBL1818218)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350951(CHEMBL1818209)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350950(CHEMBL1818210)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350948(CHEMBL1818217)
Affinity DataEC50:  848nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350952(CHEMBL1818215)
Affinity DataEC50:  468nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350949(CHEMBL1818214)
Affinity DataEC50:  186nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350953(CHEMBL1818213)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350954(CHEMBL1818212)
Affinity DataEC50:  581nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350955(CHEMBL1818211)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350950(CHEMBL1818210)
Affinity DataEC50:  215nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350951(CHEMBL1818209)
Affinity DataEC50:  175nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203072(3-isothiocyanatoprop-1-ene | Allyl isothiocyanate ...)
Affinity DataEC50:  5.81E+3nMAssay Description:Agonist activity at rat TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50203072(3-isothiocyanatoprop-1-ene | Allyl isothiocyanate ...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50350949(CHEMBL1818214)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as calcium influx measured at every 1 second for 60 seconds by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed