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Found 10 Enz. Inhib. hit(s) with all data for entry = 5105
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85134(Isofagomine derivative, 7)
Affinity DataKi:  0.0700nMpH: 7.0Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85134(Isofagomine derivative, 7)
Affinity DataKi:  0.200nMpH: 5.5Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM50075408(5-(hydroxymethyl)piperidine-3,4-diol | CHEMBL34512...)
Affinity DataKi:  5nMpH: 7.0Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM50075408(5-(hydroxymethyl)piperidine-3,4-diol | CHEMBL34512...)
Affinity DataKi:  23nMpH: 5.5Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85133(Isofagomine derivative, 10)
Affinity DataKi:  100nMpH: 5.5Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85133(Isofagomine derivative, 10)
Affinity DataKi:  110nMpH: 7.0Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85131(Isofagomine derivative, 6)
Affinity DataKi:  210nMpH: 7.0Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85132(Isofagomine derivative, 8)
Affinity DataKi:  600nMpH: 5.5Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85131(Isofagomine derivative, 6)
Affinity DataKi:  610nMpH: 5.5Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
University of British Columbia

LigandPNGBDBM85132(Isofagomine derivative, 8)
Affinity DataKi:  1.40E+3nMpH: 7.0Assay Description:Fluorescene-based assay using beta-glucocerebrosidase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed