Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50035853
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014005(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  15nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014007(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  69nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014009(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  505nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014013(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  603nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014012(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  913nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014004(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014011(4-Ethyl-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dica...)
Affinity DataKi:  1.01E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014008(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  1.05E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014010(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  2.09E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014006(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  4.41E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKi:  7.33E+4nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed