Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 5436
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86341BDBM86341(Phosphodiester analog, 4j (S4A) | Phosphodiester a...)
Affinity DataIC50: 17nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86345BDBM86345(Phosphodiester analog, 6(S4A) | Phosphodiester ana...)
Affinity DataIC50: 30nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86339BDBM86339(Phosphodiester analog, 4h)
Affinity DataIC50: 55nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86342BDBM86342(Phosphodiester analog, 4k)
Affinity DataIC50: 100nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86340BDBM86340(Phosphodiester analog, 4i)
Affinity DataIC50: 120nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86343BDBM86343(Phosphodiester analog, 4l)
Affinity DataIC50: 130nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86338BDBM86338(Phosphodiester analog, 4g)
Affinity DataIC50: 4.00E+3nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86345BDBM86345(Phosphodiester analog, 6(S4A) | Phosphodiester ana...)
Affinity DataIC50: 9.00E+3nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86329BDBM86329(Phosphodiester analog, 3j)
Affinity DataIC50: 1.10E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86337BDBM86337(Phosphodiester analog, 4f)
Affinity DataIC50: 1.10E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86341BDBM86341(Phosphodiester analog, 4j (S4A) | Phosphodiester a...)
Affinity DataIC50: 1.20E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86336BDBM86336(Phosphodiester analog, 4e)
Affinity DataIC50: 1.90E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86335BDBM86335(Phosphodiester analog, 4d)
Affinity DataIC50: 3.50E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86318BDBM86318(Phosphodiester analog, 1)
Affinity DataIC50: 3.60E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86344BDBM86344(Phosphodiester analog, 5)
Affinity DataIC50: 4.50E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86327BDBM86327(Phosphodiester analog, 3h)
Affinity DataIC50: 6.60E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86331BDBM86331(Phosphodiester analog, 3l)
Affinity DataIC50: 7.00E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86328BDBM86328(Phosphodiester analog, 3i)
Affinity DataIC50: 9.40E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86330BDBM86330(Phosphodiester analog, 3k)
Affinity DataIC50: 1.54E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86319BDBM86319(Phosphodiester analog, 2)
Affinity DataIC50: 1.74E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86324BDBM86324(Phosphodiester analog, 3e)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86325BDBM86325(Phosphodiester analog, 3f)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86322BDBM86322(Phosphodiester analog, 3c)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86323BDBM86323(Phosphodiester analog, 3d)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86326BDBM86326(Phosphodiester analog, 3g)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86332BDBM86332(Phosphodiester analog, 4a)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86333BDBM86333(Phosphodiester analog, 4b)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86320BDBM86320(Phosphodiester analog, 3a)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86321BDBM86321(Phosphodiester analog, 3b)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
National Cancer Institute-Frederick

LigandChemical structure of BindingDB Monomer ID 86334BDBM86334(Phosphodiester analog, 4c)
Affinity DataIC50: 2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed