Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50041937
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.263nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.339nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419034(CHEMBL1813321)
Affinity DataKi:  3.39nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419039(CHEMBL1813323)
Affinity DataKi:  3.98nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419040(CHEMBL1813324)
Affinity DataKi:  14.4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419035(CHEMBL1813322)
Affinity DataKi:  19.9nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419032(CHEMBL1813174)
Affinity DataKi:  20.4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419036(CHEMBL1813325)
Affinity DataKi:  36.3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419039(CHEMBL1813323)
Affinity DataKi:  40.7nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419033(CHEMBL1813319)
Affinity DataKi:  42.7nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419038(CHEMBL1813320)
Affinity DataKi:  57.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419035(CHEMBL1813322)
Affinity DataKi:  93.3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419040(CHEMBL1813324)
Affinity DataKi:  158nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419034(CHEMBL1813321)
Affinity DataKi:  182nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419041(CHEMBL1813327)
Affinity DataKi:  245nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419041(CHEMBL1813327)
Affinity DataKi:  288nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419037(CHEMBL1813326)
Affinity DataKi:  309nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419037(CHEMBL1813326)
Affinity DataKi:  380nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419036(CHEMBL1813325)
Affinity DataKi:  741nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT1 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419038(CHEMBL1813320)
Affinity DataKi:  813nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419033(CHEMBL1813319)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50419032(CHEMBL1813174)
Affinity DataKi:  2.09E+3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human cloned MT2 receptor expressed in mouse NIH-3T3 cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed