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Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50033830
TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352114(CHEMBL1824509 | CHEMBL1852788)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352114(CHEMBL1824509 | CHEMBL1852788)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352116(CHEMBL1824512 | CHEMBL1852558)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352118(CHEMBL1824513 | CHEMBL1852602)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352121(CHEMBL1824511 | CHEMBL1852555)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352119(CHEMBL1824515 | CHEMBL1852393)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352116(CHEMBL1824512 | CHEMBL1852558)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352117(CHEMBL1824514 | CHEMBL1852672)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352122(CHEMBL1824517 | CHEMBL1852458)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352120(CHEMBL1824516 | CHEMBL1852814)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352123(CHEMBL1824518 | CHEMBL1852475)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352121(CHEMBL1824511 | CHEMBL1852555)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352118(CHEMBL1824513 | CHEMBL1852602)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352123(CHEMBL1824518 | CHEMBL1852475)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352120(CHEMBL1824516 | CHEMBL1852814)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352117(CHEMBL1824514 | CHEMBL1852672)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352116(CHEMBL1824512 | CHEMBL1852558)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352119(CHEMBL1824515 | CHEMBL1852393)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352118(CHEMBL1824513 | CHEMBL1852602)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352122(CHEMBL1824517 | CHEMBL1852458)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]-norBNI from kappa opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352119(CHEMBL1824515 | CHEMBL1852393)
Affinity DataKi:  274nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352121(CHEMBL1824511 | CHEMBL1852555)
Affinity DataKi:  294nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352117(CHEMBL1824514 | CHEMBL1852672)
Affinity DataKi:  502nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352122(CHEMBL1824517 | CHEMBL1852458)
Affinity DataKi:  526nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352114(CHEMBL1824509 | CHEMBL1852788)
Affinity DataKi:  602nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352120(CHEMBL1824516 | CHEMBL1852814)
Affinity DataKi:  866nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352123(CHEMBL1824518 | CHEMBL1852475)
Affinity DataKi:  2.59E+3nMAssay Description:Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352116(CHEMBL1824512 | CHEMBL1852558)
Affinity DataEC50:  1.10nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352122(CHEMBL1824517 | CHEMBL1852458)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity against mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)
Affinity DataEC50:  1.20nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352118(CHEMBL1824513 | CHEMBL1852602)
Affinity DataEC50:  1.30nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352119(CHEMBL1824515 | CHEMBL1852393)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity against mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352120(CHEMBL1824516 | CHEMBL1852814)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity against mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352117(CHEMBL1824514 | CHEMBL1852672)
Affinity DataEC50:  2.30nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352123(CHEMBL1824518 | CHEMBL1852475)
Affinity DataEC50:  5.10nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352114(CHEMBL1824509 | CHEMBL1852788)
Affinity DataEC50:  0.830nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352121(CHEMBL1824511 | CHEMBL1852555)
Affinity DataEC50:  1.5nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed