Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50033895
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353455(CHEMBL1830049)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353456(CHEMBL1830050)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353453(CHEMBL1830047)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353458(CHEMBL1830052)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353457(CHEMBL1830051)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353452(CHEMBL1830046)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353459(CHEMBL1830053)
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353449(CHEMBL1830043)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353450(CHEMBL1830044)
Affinity DataKi:  7.80nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353454(CHEMBL1830048)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353448(CHEMBL1830042)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353451(CHEMBL1830045)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-S36057 from rat MCH1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50353448(CHEMBL1830042)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed