Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50033777
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351130(CHEMBL1817895)
Affinity DataIC50: 0.260nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351134(CHEMBL1817891)
Affinity DataIC50: 0.340nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351127(CHEMBL1817892)
Affinity DataIC50: 0.420nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50081420((7S,9R)-7-(3,5-Bis-trifluoromethyl-benzyl)-9-methy...)
Affinity DataIC50: 0.450nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351126(CHEMBL1817890)
Affinity DataIC50: 0.810nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351125(CHEMBL1817889 | CHEMBL1817897)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351125(CHEMBL1817889 | CHEMBL1817897)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351125(CHEMBL1817889 | CHEMBL1817897)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351123(CHEMBL1817887)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351128(CHEMBL1817893)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351122(CHEMBL1817886)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351124(CHEMBL1817888)
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351113(CHEMBL1817832)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351129(CHEMBL1817894)
Affinity DataIC50: 5.90nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351117(CHEMBL1817837)
Affinity DataIC50: 6.10nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351110(CHEMBL1817829)
Affinity DataIC50: 6.60nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351121(CHEMBL1817885)
Affinity DataIC50: 9.5nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351119(CHEMBL1817883)
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351131(CHEMBL1817896)
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351118(CHEMBL1817882)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351111(CHEMBL1817830)
Affinity DataIC50: 31nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351116(CHEMBL1817836)
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351120(CHEMBL1817884)
Affinity DataIC50: 55nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351112(CHEMBL1817831)
Affinity DataIC50: 77nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351109(CHEMBL1817821)
Affinity DataIC50: 97nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351107(CHEMBL1817817)
Affinity DataIC50: 97nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351108(CHEMBL1817820)
Affinity DataIC50: 97nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351115(CHEMBL1817834)
Affinity DataIC50: 220nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351114(CHEMBL1817833)
Affinity DataIC50: 270nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50351133(CHEMBL1817828)
Affinity DataIC50: 280nMAssay Description:Displacement of [125I]BH-SP from human tachykinin NK1 receptor expressed in IM9 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed