Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50039480
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22032BDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353493BDBM50353493(CHEMBL1830760)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22040BDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353499BDBM50353499(CHEMBL1830752)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353495BDBM50353495(CHEMBL1830756)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353485BDBM50353485(CHEMBL1830767)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353487BDBM50353487(CHEMBL1830764)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353492BDBM50353492(CHEMBL1830759)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353505BDBM50353505(CHEMBL1830744)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353497BDBM50353497(CHEMBL1830753)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353503BDBM50353503(CHEMBL1830748)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353491BDBM50353491(CHEMBL1830761)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353496BDBM50353496(CHEMBL1830755)
Affinity DataKi:  177nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353486BDBM50353486(CHEMBL1830766)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353502BDBM50353502(CHEMBL1830747)
Affinity DataKi:  267nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353501BDBM50353501(CHEMBL1830751)
Affinity DataKi:  346nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353517BDBM50353517(CHEMBL1830733)
Affinity DataKi:  379nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353510BDBM50353510(CHEMBL1830738)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353490BDBM50353490(CHEMBL1830763)
Affinity DataKi:  487nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353533BDBM50353533(CHEMBL1830743)
Affinity DataKi:  489nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353520BDBM50353520(CHEMBL1830727)
Affinity DataKi:  613nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353512BDBM50353512(CHEMBL1830737)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353516BDBM50353516(CHEMBL1830732)
Affinity DataKi:  651nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353532BDBM50353532(CHEMBL1830757)
Affinity DataKi:  704nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353528BDBM50353528(CHEMBL1830719)
Affinity DataKi:  772nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353488BDBM50353488(CHEMBL1830765)
Affinity DataKi:  877nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353527BDBM50353527(CHEMBL1830720)
Affinity DataKi:  914nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353498BDBM50353498(CHEMBL1830754)
Affinity DataKi:  942nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353506BDBM50353506(CHEMBL1830745)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353494BDBM50353494(CHEMBL1830758)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353500BDBM50353500(CHEMBL1830750)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353489BDBM50353489(CHEMBL1830762)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353513BDBM50353513(CHEMBL1830735)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353530BDBM50353530(CHEMBL1830749)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353504BDBM50353504(CHEMBL1830746)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353521BDBM50353521(CHEMBL1830726)
Affinity DataKi:  3.46E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353526BDBM50353526(CHEMBL1830721)
Affinity DataKi:  4.19E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353508BDBM50353508(CHEMBL1830742)
Affinity DataKi:  4.34E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353519BDBM50353519(CHEMBL1830728)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353525BDBM50353525(CHEMBL1830722)
Affinity DataKi:  4.87E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353518BDBM50353518(CHEMBL1830729)
Affinity DataKi:  5.49E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353511BDBM50353511(CHEMBL1830739)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353515BDBM50353515(CHEMBL1830734)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353509BDBM50353509(CHEMBL1830740)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353524BDBM50353524(CHEMBL1830723)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353529BDBM50353529(CHEMBL1830718)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353514BDBM50353514(CHEMBL1830736)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353531BDBM50353531(CHEMBL1830731)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353535BDBM50353535(CHEMBL1830717)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50353534BDBM50353534(CHEMBL1830730)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2013
Entry Details Article
PubMed
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