Compile Data Set for Download or QSAR
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Found 20 Enz. Inhib. hit(s) with all data for entry = 50033905
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353649(CHEMBL1829835)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353651(CHEMBL1829841)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353653(CHEMBL1829843)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353652(CHEMBL1829842)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353647(CHEMBL1829832)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353654(CHEMBL1829822)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of PKCzeta in human U937 cells assessed as inhibition of TNFalpha-induced NF-kB activation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353655(CHEMBL1829834)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353650(CHEMBL1829837)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50353648(CHEMBL1829833)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human PKCzeta assessed as [gamma32P]ATP utilization using myelin basic protein as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed