Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50004578
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484340BDBM50484340(CHEMBL1835512)
Affinity DataKi:  160nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484329BDBM50484329(CHEMBL1835505)
Affinity DataKi:  210nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484339BDBM50484339(CHEMBL1835509)
Affinity DataKi:  360nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484334BDBM50484334(CHEMBL1835504)
Affinity DataKi:  450nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484342BDBM50484342(CHEMBL1835511)
Affinity DataKi:  470nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484330BDBM50484330(CHEMBL1835507)
Affinity DataKi:  520nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484328BDBM50484328(CHEMBL1835503)
Affinity DataKi:  650nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484343BDBM50484343(CHEMBL1835510)
Affinity DataKi:  820nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484332BDBM50484332(CHEMBL1835514)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484337BDBM50484337(CHEMBL1835501)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484331BDBM50484331(CHEMBL1835508)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484324BDBM50484324(CHEMBL1835515)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484338BDBM50484338(CHEMBL1835506)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484325BDBM50484325(CHEMBL1835499)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484327BDBM50484327(CHEMBL1835502)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484336BDBM50484336(CHEMBL1835498)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484326BDBM50484326(CHEMBL1835500)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484341BDBM50484341(CHEMBL1835497)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484323BDBM50484323(CHEMBL1835496)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484335BDBM50484335(CHEMBL1835513)
Affinity DataKi: >2.42E+5nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Volgograd State Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50484333BDBM50484333(CHEMBL1835516)
Affinity DataKi: >2.49E+5nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed