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Found 21 Enz. Inhib. hit(s) with all data for entry = 50004578
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484340(CHEMBL1835512)
Affinity DataKi:  160nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484329(CHEMBL1835505)
Affinity DataKi:  210nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484339(CHEMBL1835509)
Affinity DataKi:  360nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484334(CHEMBL1835504)
Affinity DataKi:  450nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484342(CHEMBL1835511)
Affinity DataKi:  470nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484330(CHEMBL1835507)
Affinity DataKi:  520nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484328(CHEMBL1835503)
Affinity DataKi:  650nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484343(CHEMBL1835510)
Affinity DataKi:  820nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484332(CHEMBL1835514)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484331(CHEMBL1835508)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484324(CHEMBL1835515)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484337(CHEMBL1835501)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484338(CHEMBL1835506)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484325(CHEMBL1835499)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484327(CHEMBL1835502)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484336(CHEMBL1835498)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484326(CHEMBL1835500)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484341(CHEMBL1835497)
Affinity DataKi:  6.30E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484323(CHEMBL1835496)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484335(CHEMBL1835513)
Affinity DataKi: >2.42E+5nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Volgograd State Medical University

Curated by ChEMBL
LigandPNGBDBM50484333(CHEMBL1835516)
Affinity DataKi: >2.49E+5nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 reverse transcriptase p66/p51 heterodimer using [8-3H]dGTP as substrate after 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed